SCHEMBL4733913

SCHEMBL4733913

O=C(c1ccncn1)N(Cc1ccc(Cl)nc1)c1ccc(F)cc1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDK1 Q15118 5/20 0.43
MAPK14 Q16539 2/20 0.43
BCL2A1 Q16548 1/20 0.40
CXCR2 P25025 1/20 0.38
P2RX7 Q99572 1/20 0.37
KCNQ3 O43525 1/20 0.36
KCNQ2 O43526 1/20 0.36
KCNE1 P15382 1/20 0.36
KCNQ1 P51787 1/20 0.36
BACE1 P56817 1/20 0.36
HSP90AA1 P07900 1/20 0.35
HSP90AB1 P08238 1/20 0.35
PDK2 Q15119 1/20 0.35
PDK3 Q15120 1/20 0.35
PDK4 Q16654 1/20 0.35
ALDH1A1 P00352 1/20 0.34
MDM2 Q00987 1/20 0.34
F2 P00734 1/20 0.34
QPCT Q16769 1/20 0.34
GAA P10253 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4734214 0.85 MAPK14 (0.43) PDK1MAPK14BCL2A1CXCR2HSP90AA1
SCHEMBL4784324 0.85 PDK1 (0.46) PDK1MAPK14BCL2A1CXCR2ALDH1A1
SCHEMBL4738782 0.83 MAPK14 (0.45) PDK1MAPK14BCL2A1CXCR2KCNQ3
SCHEMBL4737107 0.80 GAA (0.58) PDK1MAPK14BCL2A1CXCR2GAA
SCHEMBL3822748 0.79 BCL2A1 (0.52) PDK1MAPK14BCL2A1CXCR2KCNQ3
SCHEMBL4737244 0.79 ME2 (0.41) MAPK14CXCR2ALDH1A1TSHR
SCHEMBL3066549 0.78 BCL2A1 (0.47) PDK1MAPK14BCL2A1KCNQ3KCNQ2
SCHEMBL3071604 0.75 BCL2A1 (0.44) PDK1BCL2A1KCNQ3KCNQ2KCNE1
SCHEMBL3065683 0.73 BCL2A1 (0.42) PDK1BCL2A1KCNQ3KCNQ2KCNE1
SCHEMBL8193274 0.70 MAPK14 (0.42) PDK1MAPK14CXCR2P2RX7HSP90AA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008073461-A2 ION CHANNEL MODULATORS WYETH (US) 2008-06-19 WO claimed