SCHEMBL4734701

SCHEMBL4734701

C=CCc1c(C(=O)OCC)cc2c(nc(C)n2C)c1OC(=O)C(C)(C)C

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.38
CYP3A4 P08684 1/20 0.36
CYP2C19 P33261 1/20 0.36
KDM4E B2RXH2 7/20 0.34
HSD17B10 Q99714 4/20 0.34
KMT2A Q03164 3/20 0.34
ELANE P08246 2/20 0.32
PRTN3 P24158 1/20 0.32
L3MBTL1 Q9Y468 1/20 0.32
RXRA P19793 1/20 0.32
MEN1 O00255 1/20 0.32
RAB9A P51151 1/20 0.32
HPGD P15428 4/20 0.31
GAA P10253 3/20 0.31
GLA P06280 2/20 0.31
HIF1A Q16665 2/20 0.31
CASP1 P29466 1/20 0.31
CASP7 P55210 1/20 0.31
POLB P06746 1/20 0.31
STAT6 P42226 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4737618 0.91 CYP3A4 (0.36) ALDH1A1CYP3A4CYP2C19KDM4EHSD17B10
SCHEMBL4735693 0.83 CYP3A4 (0.37) CYP3A4CYP2C19ELANEPRTN3SIRT2
SCHEMBL4737295 0.81 ALDH1A1 (0.37) ALDH1A1CYP3A4CYP2C19KDM4EHSD17B10
SCHEMBL4737293 0.81 ALDH1A1 (0.37) ALDH1A1CYP3A4CYP2C19KDM4EHSD17B10
SCHEMBL4737617 0.79 TSHR (0.33) ALDH1A1CYP2C19KMT2AMEN1TSHR
SCHEMBL4739265 0.77
SCHEMBL4739250 0.70 ALDH1A1 (0.43) ALDH1A1KDM4EHSD17B10KMT2AL3MBTL1
SCHEMBL4739806 0.69 HSP90AA1 (0.34) ALDH1A1KDM4EHSD17B10KMT2AELANE
SCHEMBL4738360 0.69
SCHEMBL5116642 0.68 GAA (0.43) ALDH1A1KDM4EHSD17B10KMT2AL3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008071765-A1 PHARMACEUTICALLY ACTIVE SPIRO-SUBSTITUTED BENZIMIDAZOLE DERIVATIVES NYCOMED GMBH (DE) 2008-06-19 WO disclosed