SCHEMBL4737293

SCHEMBL4737293

CCOC(=O)c1cc2c(nc(C)n2C)c(OC(=O)C(C)(C)C)c1C/C=C1\CCc2ccccc21

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.37
HPGD P15428 4/20 0.37
KDM4E B2RXH2 3/20 0.37
TDP1 Q9NUW8 1/20 0.37
L3MBTL1 Q9Y468 1/20 0.37
ELANE P08246 1/20 0.34
PRTN3 P24158 1/20 0.34
POLB P06746 3/20 0.32
HSP90AA1 P07900 2/20 0.32
MAPT P10636 2/20 0.32
HSP90AB1 P08238 1/20 0.32
HSD17B10 Q99714 1/20 0.32
KMT2A Q03164 2/20 0.32
MEN1 O00255 1/20 0.31
USP2 O75604 1/20 0.31
TSHR P16473 1/20 0.31
RAB9A P51151 1/20 0.31
GABRP O00591 1/20 0.31
GABRD O14764 1/20 0.31
GABRA1 P14867 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4737295 1.00 ALDH1A1 (0.37) ALDH1A1HPGDKDM4ETDP1L3MBTL1
SCHEMBL4737617 0.91 TSHR (0.33) ALDH1A1KMT2AMEN1TSHRGABRP
SCHEMBL4736255 0.88 ALDH1A1 (0.39) ALDH1A1HPGDKDM4ETDP1L3MBTL1
SCHEMBL4737618 0.82 CYP3A4 (0.36) ALDH1A1HPGDKDM4EL3MBTL1ELANE
SCHEMBL4736286 0.81
SCHEMBL4734701 0.81 ALDH1A1 (0.38) ALDH1A1HPGDKDM4EL3MBTL1ELANE
SCHEMBL4735242 0.80 FNTA (0.31)
SCHEMBL4735621 0.80
SCHEMBL4735019 0.79 NQO2 (0.38) MAPTTP53
SCHEMBL4738139 0.78 ACHE (0.35) ALDH1A1HPGDKDM4EMAPTKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008071765-A1 PHARMACEUTICALLY ACTIVE SPIRO-SUBSTITUTED BENZIMIDAZOLE DERIVATIVES NYCOMED GMBH (DE) 2008-06-19 WO disclosed