SCHEMBL4734706

SCHEMBL4734706

CCc1ccccc1-c1ccc(S(=O)(=O)NC2CCN(C(=O)OC(C)(C)C)CC2)c(C(F)(F)F)c1

nearest known ligand 0.55

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
SFRP1 Q8N474 10/20 0.55
BRD4 O60885 2/20 0.53
CCR8 P51685 1/20 0.50
WNT3 P56703 5/20 0.49
NR1H2 P55055 1/20 0.47
GPR119 Q8TDV5 1/20 0.46
EPHX2 P34913 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4884331 0.93 SFRP1 (0.53) SFRP1BRD4CCR8WNT3NR1H2
SCHEMBL4736053 0.90 SFRP1 (0.57) SFRP1BRD4CCR8WNT3NR1H2
SCHEMBL4734276 0.90 SFRP1 (0.57) SFRP1BRD4CCR8WNT3NR1H2
SCHEMBL4734372 0.90 SFRP1 (0.57) SFRP1BRD4CCR8WNT3NR1H2
SCHEMBL4735311 0.89 SFRP1 (0.51) SFRP1WNT3
SCHEMBL4846943 0.89 SFRP1 (0.56) SFRP1BRD4CCR8WNT3NR1H2
SCHEMBL4735770 0.88 SFRP1 (0.55) SFRP1BRD4CCR8WNT3NR1H2
SCHEMBL4799560 0.87 SFRP1 (0.62) SFRP1BRD4CCR8WNT3NR1H2
SCHEMBL4733043 0.87 SFRP1 (0.55) SFRP1BRD4CCR8WNT3NR1H2
SCHEMBL4734592 0.87 SFRP1 (0.55) SFRP1BRD4CCR8WNT3NR1H2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008061016-A1 N-SUBSTITUTED PIPERIDINYL 4 -ARYLSULFONAMIDES AS MODULATORS OF THE SECRETED FRIZZLED RELATED PROTEIN- 1 WYETH (US) 2008-05-22 WO disclosed