SCHEMBL4735459

SCHEMBL4735459

COc1c(C)cc(C(=O)c2ccc(Cl)nc2)cc1C

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TUBB4A P04350 2/20 0.49
TUBB P07437 2/20 0.49
TUBA3C P0DPH7 2/20 0.49
TUBA1B P68363 2/20 0.49
TUBA4A P68366 2/20 0.49
TUBB4B P68371 2/20 0.49
TUBB3 Q13509 2/20 0.49
TUBB2A Q13885 2/20 0.49
TUBB8 Q3ZCM7 2/20 0.49
TUBA3E Q6PEY2 2/20 0.49
TUBA1A Q71U36 2/20 0.49
TUBA1C Q9BQE3 2/20 0.49
TUBB6 Q9BUF5 2/20 0.49
TUBB2B Q9BVA1 2/20 0.49
TUBB1 Q9H4B7 2/20 0.49
NAPRT Q6XQN6 1/20 0.47
KCNQ3 O43525 4/20 0.47
KCNQ2 O43526 4/20 0.47
DGAT1 O75907 2/20 0.44
RAB9A P51151 3/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL38665425 0.80 HPGD (0.61) TUBB4ATUBBTUBA3CTUBA1BTUBA4A
SCHEMBL11435411 0.79 TUBB4A (0.54) TUBB4ATUBBTUBA3CTUBA1BTUBA4A
SCHEMBL7440808 0.79 NAPRT (0.72) NAPRTKCNQ3KCNQ2DGAT1RAB9A
SCHEMBL15067437 0.78 RXFP1 (0.65) TUBB4ATUBBTUBA3CTUBA1BTUBA4A
SCHEMBL10392725 0.78 CYP1A2 (0.67) NAPRTKCNQ3KCNQ2L3MBTL1TDP1
SCHEMBL17676098 0.76 RAB9A (0.64) NAPRTKCNQ3KCNQ2DGAT1RAB9A
SCHEMBL4739273 0.76 TUBB4A (0.45) TUBB4ATUBBTUBA3CTUBA1BTUBA4A
SCHEMBL16460859 0.75 KCNQ3 (0.64) KCNQ3KCNQ2MEN1KMT2AL3MBTL1
SCHEMBL10633373 0.75 NAPRT (0.53) NAPRTKCNQ3KCNQ2DGAT1RAB9A
SCHEMBL11576801 0.74 TUBB4A (0.70) TUBB4ATUBBTUBA3CTUBA1BTUBA4A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008070014-A2 BIARYL KETONE-SUBSTITUTED PIPERIDINES NEUROGEN CORPORATION (US) 2008-06-12 WO disclosed
WO-2008070014-A2 BIARYL KETONE-SUBSTITUTED PIPERIDINES NEUROGEN CORPORATION (US) 2008-06-12 WO disclosed