SCHEMBL473595

SCHEMBL473595

O=C(O)c1cccnc1-c1cccc(C(F)(F)F)c1

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.59
TDP1 Q9NUW8 2/20 0.59
LMNA P02545 2/20 0.59
MEN1 O00255 1/20 0.59
GMNN O75496 1/20 0.59
TTR P02766 1/20 0.59
CYP1A2 P05177 1/20 0.59
CYP3A4 P08684 1/20 0.59
CYP2C9 P11712 1/20 0.59
PKM P14618 1/20 0.59
NFKB1 P19838 1/20 0.59
UGT1A1 P22309 1/20 0.59
PTGS1 P23219 1/20 0.59
PTGS2 P35354 1/20 0.59
PMP22 Q01453 1/20 0.59
DHODH Q02127 1/20 0.59
KMT2A Q03164 1/20 0.59
TEAD4 Q15561 1/20 0.59
HIF1A Q16665 1/20 0.59
GPR35 Q9HC97 1/20 0.59

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9002267 0.90 RORB (0.56) ALDH1A1TDP1LMNAMEN1GMNN
SCHEMBL5178386 0.87 PARP1 (0.58) ALDH1A1TDP1LMNAMEN1GMNN
SCHEMBL29978735 0.84 TDP1 (0.61) ALDH1A1TDP1LMNAMEN1GMNN
SCHEMBL4197626 0.84 TDP1 (0.61) ALDH1A1TDP1LMNAMEN1GMNN
Hydrochloric Acid SCHEMBL6201867 0.82 KDM4E (0.59) ALDH1A1TDP1LMNAMEN1GMNN
SCHEMBL3345499 0.81 KMO (0.56) ALDH1A1TDP1LMNAMEN1GMNN
SCHEMBL5125812 0.80 KDM4E (0.65) ALDH1A1TDP1LMNACYP3A4DHODH
SCHEMBL8936334 0.78 ADORA2A (0.51) ALDH1A1MEN1KMT2AKDM4EKMO
SCHEMBL912675 0.78 KDM4E (0.77) ALDH1A1TDP1LMNAMEN1CYP3A4
SCHEMBL31586013 0.78 KDM4E (0.77) ALDH1A1TDP1LMNAMEN1CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2411011-A1 NOVEL AMINOPYRIDINE DERIVATIVES HAVING AURORA A SELECTIVE INHIBITORY ACTION MSD K.K. (JP) 2012-02-01 EP disclosed
WO-2010111056-A1 NOVEL AMINOPYRIDINE DERIVATIVES HAVING AURORA A SELECTIVE INHIBITORY ACTION BANYU PHARMACEUTICAL CO., LTD. (JP) 2010-09-30 WO disclosed