SCHEMBL3345499

SCHEMBL3345499

O=C(O)c1nccnc1-c1cccc(C(F)(F)F)c1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMO O15229 2/20 0.56
PIN1 Q13526 1/20 0.53
NPC1 O15118 1/20 0.52
ATM Q13315 1/20 0.52
POLB P06746 1/20 0.48
ALDH1A1 P00352 3/20 0.47
SMN1; SMN2 Q16637 1/20 0.47
XDH P47989 1/20 0.47
TLR7 Q9NYK1 1/20 0.46
TDO2 P48775 1/20 0.46
KCNA5 P22460 3/20 0.45
KCNH2 Q12809 1/20 0.45
KMT2A Q03164 3/20 0.45
ADORA2A P29274 1/20 0.45
ADORA1 P30542 1/20 0.45
RORC P51449 1/20 0.44
RORB Q92753 1/20 0.44
MEN1 O00255 2/20 0.44
IP6K1 Q92551 1/20 0.44
IP6K3 Q96PC2 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL473595 0.81 ALDH1A1 (0.59) KMOPIN1POLBALDH1A1SMN1; SMN2
SCHEMBL27827780 0.81 KMO (0.54) KMOPIN1NPC1ATMPOLB
SCHEMBL8400098 0.78 PIN1 (0.52) KMOPIN1NPC1POLBALDH1A1
SCHEMBL8936345 0.78 KMO (0.54) KMOPIN1ALDH1A1SMN1; SMN2XDH
SCHEMBL1340669 0.77 KDM4E (0.53) PIN1ATMALDH1A1SMN1; SMN2KDM4E
SCHEMBL319166 0.77 MCL1 (0.46) KMOATMPOLBALDH1A1KMT2A
SCHEMBL2057011 0.77 KMO (0.52) KMOPIN1ALDH1A1KMT2AMEN1
SCHEMBL14149905 0.77 ATM (0.60) KMONPC1ATMALDH1A1KDM4E
SCHEMBL9002267 0.77 RORB (0.56) KMOPOLBALDH1A1TDO2KCNA5
SCHEMBL7673510 0.75 MAPK14 (0.57) NPC1TDO2KCNA5KCNH2ADORA2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-102164896-A Phenethylamide derivatives and their heterocyclic analogues ACTELION PHARMACEUTICALS LTD 2011-08-24 CN claimed
WO-2010044054-A1 PHENETHYLAMIDE DERIVATIVES AND THEIR HETEROCYCLIC ANALOGUES ACTELION PHARMACEUTICALS LTD (CH) 2010-04-22 WO claimed
CN-102164896-A Phenethylamide derivatives and their heterocyclic analogues ACTELION PHARMACEUTICALS LTD 2011-08-24 CN disclosed
WO-2010044054-A1 PHENETHYLAMIDE DERIVATIVES AND THEIR HETEROCYCLIC ANALOGUES ACTELION PHARMACEUTICALS LTD (CH) 2010-04-22 WO disclosed