SCHEMBL4736200

SCHEMBL4736200

O=C(c1cccnc1)N(Cc1ccc(N2CCC(N3CCOCC3)CC2)nc1)c1ccc(F)cc1

nearest known ligand 0.44

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
PDK1 Q15118 3/20 0.44
GAA P10253 1/20 0.43
TSHR P16473 1/20 0.43
CYP3A4 P08684 2/20 0.43
CYP2D6 P10635 2/20 0.43
CYP2C9 P11712 2/20 0.43
CYP2C19 P33261 2/20 0.43
CYP1A2 P05177 1/20 0.43
CD38 P28907 1/20 0.41
SMO Q99835 1/20 0.39
AOC3 Q16853 1/20 0.38
CXCR3 P49682 1/20 0.38
ADRA1A P35348 1/20 0.38
HRH3 Q9Y5N1 1/20 0.38
KDM4E B2RXH2 2/20 0.37
MAPK14 Q16539 1/20 0.37
ALDH1A1 P00352 1/20 0.37
NAMPT P43490 1/20 0.37
MLNR O43193 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4784137 0.92 PDK1 (0.50) PDK1GAATSHRAOC3KDM4E
SCHEMBL4733572 0.89 TSHR (0.45) PDK1GAATSHRSMOCXCR3
SCHEMBL4737958 0.87 TSHR (0.48) PDK1GAATSHRCYP3A4CYP2C9
SCHEMBL4735235 0.86 GAA (0.47) PDK1GAATSHRCYP3A4CYP2C9
SCHEMBL4736742 0.85 GAA (0.46) PDK1GAATSHRCYP3A4CYP2C9
SCHEMBL4735150 0.84 TSHR (0.51) PDK1GAATSHRAOC3KDM4E
SCHEMBL4738289 0.84 GAA (0.45) PDK1GAATSHRCYP3A4CYP2C9
SCHEMBL4786168 0.84 TSHR (0.47) PDK1GAATSHRSMOKDM4E
SCHEMBL4738239 0.83 TSHR (0.49) PDK1GAATSHRKDM4EMAPK14
SCHEMBL4739086 0.83 TSHR (0.52) PDK1GAATSHRCYP3A4CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008073461-A2 ION CHANNEL MODULATORS WYETH (US) 2008-06-19 WO claimed