SCHEMBL4738239

SCHEMBL4738239

CN1CCN(c2ccc(CN(C(=O)c3cccnc3)c3ccc(F)cc3)cn2)CC1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 2/20 0.49
GAA P10253 1/20 0.49
HTT P42858 1/20 0.43
CXCR2 P25025 1/20 0.42
MAPK14 Q16539 1/20 0.41
KCNH2 Q12809 2/20 0.41
OPRM1 P35372 2/20 0.41
OPRD1 P41143 1/20 0.41
PDK1 Q15118 3/20 0.41
PTGDR2 Q9Y5Y4 1/20 0.41
SLC1A3 P43003 1/20 0.41
SLC1A2 P43004 1/20 0.41
SLC1A1 P43005 1/20 0.41
KDM4E B2RXH2 1/20 0.40
ALDH1A1 P00352 1/20 0.40
OPRK1 P41145 1/20 0.39
ME2 P23368 1/20 0.39
ME1 P48163 1/20 0.39
ME3 Q16798 1/20 0.39
EP300 Q09472 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4736729 0.96 TSHR (0.46) TSHRGAAHTTCXCR2MAPK14
SCHEMBL4737126 0.92 TSHR (0.48) TSHRGAAHTTCXCR2MAPK14
SCHEMBL4736584 0.91 TSHR (0.51) TSHRGAAHTTCXCR2MAPK14
SCHEMBL4739086 0.91 TSHR (0.52) TSHRGAAHTTCXCR2MAPK14
SCHEMBL4735150 0.91 TSHR (0.51) TSHRGAAHTTCXCR2MAPK14
SCHEMBL3830332 0.91 MEN1 (0.45) TSHRGAACXCR2MAPK14OPRM1
SCHEMBL4736483 0.90 TSHR (0.47) TSHRGAACXCR2MAPK14KCNH2
SCHEMBL4736473 0.90 OPRM1 (0.41) TSHRCXCR2MAPK14OPRM1KDM4E
SCHEMBL4735615 0.90 MAPK14 (0.45) TSHRCXCR2MAPK14OPRM1OPRD1
SCHEMBL4784137 0.89 PDK1 (0.50) TSHRGAAHTTCXCR2MAPK14

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008073461-A2 ION CHANNEL MODULATORS WYETH (US) 2008-06-19 WO claimed