SCHEMBL4736644

SCHEMBL4736644

O=C(CC1CCCN(S(=O)(=O)c2ccc3ccccc3c2)C1)NN1CC2CCCC2C1

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AKR1C3 P42330 4/20 0.59
EIF2AK3 Q9NZJ5 1/20 0.59
AKR1C1 Q04828 1/20 0.53
HDAC3 O15379 1/20 0.52
HDAC4 P56524 1/20 0.52
HDAC1 Q13547 1/20 0.52
HDAC7 Q8WUI4 1/20 0.52
HDAC2 Q92769 1/20 0.52
HDAC10 Q969S8 1/20 0.52
HDAC11 Q96DB2 1/20 0.52
HDAC8 Q9BY41 1/20 0.52
HDAC6 Q9UBN7 1/20 0.52
HDAC9 Q9UKV0 1/20 0.52
HDAC5 Q9UQL6 1/20 0.52
MCOLN3 Q8TDD5 3/20 0.50
TSHR P16473 1/20 0.50
LMNA P02545 2/20 0.49
HTT P42858 2/20 0.47
GAA P10253 1/20 0.47
NPSR1 Q6W5P4 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4739899 0.91 AKR1C3 (0.60) AKR1C3EIF2AK3AKR1C1HDAC3HDAC4
SCHEMBL4739818 0.91 AKR1C3 (0.60) AKR1C3EIF2AK3AKR1C1HDAC3HDAC4
SCHEMBL4737612 0.87 LMNA (0.50) AKR1C3AKR1C1HDAC3HDAC4HDAC1
SCHEMBL4736646 0.84 AKR1C3 (0.52) AKR1C3EIF2AK3AKR1C1HDAC3HDAC4
SCHEMBL4737423 0.83 CYP3A4 (0.65) LMNAHTTGAANPSR1MEN1
SCHEMBL4736821 0.82 HDAC3 (0.51) HDAC3HDAC4HDAC1HDAC7HDAC2
SCHEMBL4741684 0.81 ALDH1A1 (0.49) LMNAMEN1KMT2APKM
SCHEMBL4736785 0.81 HDAC3 (0.51) AKR1C3AKR1C1HDAC3HDAC4HDAC1
SCHEMBL4782857 0.79 POLB (0.47) AKR1C3EIF2AK3AKR1C1HDAC3HDAC4
SCHEMBL12939736 0.79 AKR1C3 (0.63) AKR1C3EIF2AK3AKR1C1HDAC3HDAC4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008087654-A2 PIPERIDINES AS INHIBITORS OF 11β-HYDROXYSTEROID DEHYDROGENASE TYPE 1 CADILA HEALTHCARE LIMITED (IN) 2008-07-24 WO claimed
WO-2008087654-A2 PIPERIDINES AS INHIBITORS OF 11β-HYDROXYSTEROID DEHYDROGENASE TYPE 1 CADILA HEALTHCARE LIMITED (IN) 2008-07-24 WO disclosed