SCHEMBL4736797

SCHEMBL4736797

CSc1nc2c(c(-c3ccc(Cl)cc3)n1)-c1ccccc1CC2

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TYMS P04818 6/20 0.43
KDM4E B2RXH2 3/20 0.43
CCNA2 P20248 2/20 0.42
CDK2 P24941 2/20 0.42
ADORA2A P29274 1/20 0.38
ADORA1 P30542 1/20 0.38
HRH1 P35367 1/20 0.38
HRH4 Q9H3N8 1/20 0.38
ALDH1A1 P00352 3/20 0.36
LMNA P02545 2/20 0.36
TDP1 Q9NUW8 2/20 0.36
HPGD P15428 2/20 0.36
NPC1 O15118 2/20 0.36
MAPT P10636 2/20 0.36
ALOX12 P18054 1/20 0.36
POLB P06746 1/20 0.36
L3MBTL1 Q9Y468 1/20 0.36
NPSR1 Q6W5P4 2/20 0.35
RAB9A P51151 1/20 0.35
KMT2A Q03164 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4787503 0.78 PTGS2 (0.42) TYMSKDM4EADORA2AADORA1HRH1
SCHEMBL4741269 0.74 ADORA1 (0.45) KDM4ECCNA2CDK2ADORA1HRH1
SCHEMBL4839488 0.72 KDM4E (0.57) KDM4EADORA2AADORA1ALDH1A1LMNA
SCHEMBL17279668 0.69 TYMS (0.41) TYMSHRH1HRH4ALDH1A1TDP1
SCHEMBL4841960 0.67 KDM4E (0.51) KDM4EALDH1A1LMNATDP1NPC1
SCHEMBL8326420 0.66 CCNA2 (0.67) CCNA2CDK2
SCHEMBL4739911 0.66 TYMS (0.52) TYMSADORA2AADORA1
SCHEMBL7513198 0.65 KDM4E (0.59) KDM4ECCNA2CDK2ALDH1A1LMNA
SCHEMBL25603965 0.65 NPSR1 (0.63) KDM4EALDH1A1LMNAHPGDNPC1
SCHEMBL10812119 0.64 NPSR1 (0.68) KDM4EADORA2AADORA1ALDH1A1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008086158-A1 BENZODIHYDROQUINAZOLINE AS PI3 KINASE INHIBITORS SMITHKLINE BEECHAM CORPORATION (US) 2008-07-17 WO disclosed
WO-2008086158-A1 BENZODIHYDROQUINAZOLINE AS PI3 KINASE INHIBITORS SMITHKLINE BEECHAM CORPORATION (US) 2008-07-17 WO disclosed