SCHEMBL4737022

SCHEMBL4737022

COC(=O)N1CCN(C2CNC2)CC1

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CHRNB2 P17787 3/20 0.55
CHRNA4 P43681 3/20 0.55
CHRNB4 P30926 2/20 0.55
CHRNA3 P32297 2/20 0.55
L3MBTL1 Q9Y468 1/20 0.39
IRAK4 Q9NWZ3 5/20 0.38
MAPT P10636 2/20 0.38
KMT2A Q03164 2/20 0.38
ALDH1A1 P00352 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.36
ACACB O00763 2/20 0.36
ACACA Q13085 2/20 0.36
USP2 O75604 1/20 0.36
CYP1A2 P05177 1/20 0.36
CYP2C9 P11712 1/20 0.36
PKM P14618 1/20 0.36
CHRNA7 P36544 1/20 0.35
HRH3 Q9Y5N1 1/20 0.35
CCNC P24863 1/20 0.35
CDK8 P49336 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL4737835 0.98 CHRNB2 (0.53) CHRNB2CHRNA4CHRNB4CHRNA3L3MBTL1
SCHEMBL1306212 0.81 USP2 (0.49) L3MBTL1MAPTKMT2AALDH1A1SMN1; SMN2
Hydrochloric Acid SCHEMBL7811769 0.80 USP2 (0.47) L3MBTL1MAPTKMT2AALDH1A1SMN1; SMN2
SCHEMBL6840205 0.79 CHRNB2 (0.50) CHRNB2CHRNA4CHRNB4CHRNA3IRAK4
SCHEMBL23334495 0.78 POLB (0.57) KMT2AALDH1A1PKMHRH3
SCHEMBL21482489 0.78 POLB (0.57) KMT2AALDH1A1PKMHRH3
SCHEMBL3772648 0.77 MAPT (0.40) IRAK4MAPTKMT2AALDH1A1ACACB
Hydrochloric Acid SCHEMBL5327246 0.77 CHRNB2 (0.48) CHRNB2CHRNA4CHRNB4CHRNA3IRAK4
Hydrochloric Acid SCHEMBL3760127 0.77 CHRNB2 (0.48) CHRNB2CHRNA4CHRNB4CHRNA3IRAK4
SCHEMBL20617537 0.77 L3MBTL1 (0.53) CHRNB2CHRNA4CHRNB4CHRNA3L3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008076042-A1 AZETIDINPIPERAZINE DERIVATIVES THAT ARE NEUROKININ (NK) RECEPTOR ANTAGONISTS AND THEIR USE. ASTRAZENECA AB (SE) 2008-06-26 WO disclosed