SCHEMBL4737261

SCHEMBL4737261

CC(C)c1ccc2c(c1)C(=O)Cc1ccc(F)cc1S2

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 1/20 0.44
OPRK1 P41145 1/20 0.44
PDE4D Q08499 1/20 0.44
HPGD P15428 4/20 0.43
KMT2A Q03164 4/20 0.43
ALDH1A1 P00352 3/20 0.43
MEN1 O00255 3/20 0.43
LMNA P02545 2/20 0.43
MAPT P10636 1/20 0.43
L3MBTL1 Q9Y468 1/20 0.43
KDM4E B2RXH2 2/20 0.40
BLM P54132 1/20 0.37
HTT P42858 1/20 0.37
ATM Q13315 1/20 0.37
GFER P55789 1/20 0.37
HSD17B10 Q99714 1/20 0.37
CYP17A1 P05093 1/20 0.33
ACHE P22303 1/20 0.33
DRD2 P14416 1/20 0.32
MAOA P21397 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11401676 0.87 PTGS2 (0.63) PTGS2OPRK1PDE4DHPGDKMT2A
SCHEMBL11397123 0.86 PTGS2 (0.50) PTGS2OPRK1PDE4DHPGDKMT2A
SCHEMBL4734664 0.82 CYP17A1 (0.39) PTGS2OPRK1PDE4DHPGDKMT2A
SCHEMBL11343598 0.80 MEN1 (0.68) PTGS2OPRK1PDE4DHPGDKMT2A
SCHEMBL11342050 0.80 ALDH1A1 (0.46) PTGS2OPRK1PDE4DHPGDKMT2A
SCHEMBL11759198 0.80 ALDH1A1 (0.56) PTGS2OPRK1PDE4DHPGDKMT2A
SCHEMBL11346578 0.79 MAPK14 (0.43) HPGDKMT2AALDH1A1MEN1LMNA
SCHEMBL11395551 0.78 PTGS2 (0.71) PTGS2OPRK1PDE4DHPGDKMT2A
SCHEMBL11759541 0.77 HPGD (0.63) PTGS2OPRK1PDE4DHPGDKMT2A
SCHEMBL11394759 0.77 PTGS2 (0.57) PTGS2OPRK1PDE4DHPGDKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008061029-A1 ARYL SULFONAMIDE DERIVATIVES AND METHODS OF THEIR USE WYETH (US) 2008-05-22 WO disclosed
US-4243805-A 3 Fluoro-10-piperazino-8-substituted 10,11-dihydrodibenzo-(bf) thiepins and method for the preparation thereof SPOFA, SPOJENE PODNIKY PRO ZDRAVOTNICKOU VYROBU (CS) 1981-01-06 US disclosed