SCHEMBL4737438

SCHEMBL4737438

Nc1nc2c(c(-c3ccc4[nH]ccc4c3)n1)-c1ccc(Br)cc1CC2

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TYMS P04818 3/20 0.47
AHR P35869 2/20 0.42
CYP2A6 P11509 1/20 0.42
NR4A2 P43354 1/20 0.42
MAP3K14 Q99558 1/20 0.36
ADORA2A P29274 2/20 0.36
ADORA1 P30542 2/20 0.36
CYP3A4 P08684 1/20 0.35
CYP2D6 P10635 1/20 0.35
MAP3K11 Q16584 1/20 0.35
NISCH Q9Y2I1 1/20 0.34
LRRK2 Q5S007 1/20 0.34
CSNK1D P48730 1/20 0.34
MAPK11 Q15759 1/20 0.34
MAPK14 Q16539 1/20 0.34
ATR Q13535 1/20 0.34
NPC1 O15118 1/20 0.34
PIK3CD O00329 2/20 0.34
ABL1 P00519 2/20 0.34
EGFR P00533 2/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4737419 0.85 MAP3K11 (0.38) ADORA2AADORA1CYP3A4CYP2D6MAP3K11
SCHEMBL6651001 0.74 TYMS (0.59) TYMSPARP10PARP11
SCHEMBL846923 0.71 BRD4 (0.47) ADORA2AADORA1CYP3A4CYP2D6MAP3K11
SCHEMBL4737435 0.69 TYMS (0.47) TYMSMAP3K14CSNK1DKDR
SCHEMBL4787500 0.66 TYMS (0.50) TYMSADORA2AADORA1
SCHEMBL4739911 0.65 TYMS (0.52) TYMSADORA2AADORA1
SCHEMBL27612533 0.65 PIK3CD (0.46) AHRADORA2AADORA1CYP3A4CYP2D6
SCHEMBL6648692 0.65 TYMS (1.00) TYMS
SCHEMBL3462787 0.64 AHR (0.70) AHRCYP2A6NR4A2MAP3K11NISCH
SCHEMBL74304 0.64 AHR (1.00) AHRCYP2A6NR4A2CYP3A4NPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008086158-A1 BENZODIHYDROQUINAZOLINE AS PI3 KINASE INHIBITORS SMITHKLINE BEECHAM CORPORATION (US) 2008-07-17 WO disclosed