SCHEMBL4737488

SCHEMBL4737488

CC(C)(CCn1cnc2cc(OC(=O)NN)ccc21)NC[C@H](O)c1cccc(NS(=O)(=O)c2ccccc2)c1

nearest known ligand 0.46

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
ADRB3 P13945 8/20 0.46
NR1I2 O75469 6/20 0.41
HPGD P15428 2/20 0.40
ALDH1A1 P00352 2/20 0.39
LMNA P02545 1/20 0.39
MAPT P10636 1/20 0.39
HTT P42858 1/20 0.39
L3MBTL1 Q9Y468 1/20 0.39
KMT2A Q03164 1/20 0.37
OPRM1 P35372 1/20 0.37
OPRD1 P41143 1/20 0.37
ADRA1A P35348 2/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Trifluoroacetic Acid SCHEMBL4647223 0.97 ADRB3 (0.45) ADRB3NR1I2HPGDALDH1A1LMNA
SCHEMBL1379766 0.93 ADRB3 (0.48) ADRB3NR1I2HPGDALDH1A1LMNA
SCHEMBL4640303 0.90 ADRB3 (0.47) ADRB3NR1I2HPGDALDH1A1LMNA
SCHEMBL4643457 0.90 ADRB3 (0.47) ADRB3NR1I2HPGDALDH1A1LMNA
SCHEMBL4917492 0.89 NR1I2 (0.43) ADRB3NR1I2HPGDALDH1A1KMT2A
SCHEMBL4908069 0.89 NR1I2 (0.43) ADRB3NR1I2HPGDALDH1A1KMT2A
SCHEMBL1377347 0.87 NR1I2 (0.45) ADRB3NR1I2HPGDALDH1A1KMT2A
SCHEMBL4914684 0.86 NR1I2 (0.44) ADRB3NR1I2HPGDALDH1A1KMT2A
SCHEMBL1379764 0.86 NR1I2 (0.44) ADRB3NR1I2HPGDALDH1A1KMT2A
SCHEMBL4649151 0.86 ALDH1A1 (0.47) ADRB3NR1I2HPGDALDH1A1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1943229-A1 BENZIMIDAZOLE DERIVATIVES FOR USE AS BETA-3 RECEPTOR AGONISTS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2008-07-16 EP claimed
WO-2007048842-A1 BENZIMIDAZOLE DERIVATIVES FOR USE AS BETA-3 RECEPTOR AGONISTS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2007-05-03 WO claimed