SCHEMBL4737570

SCHEMBL4737570

N=C(N)c1c(F)cccc1Cl

nearest known ligand 0.50

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
BACE1 P56817 1/20 0.50
GAA P10253 7/20 0.46
ITGB2 P05107 1/20 0.44
ICAM1 P05362 1/20 0.44
ITGAL P20701 1/20 0.44
PBRM1 Q86U86 1/20 0.43
JAK2 O60674 1/20 0.42
JAK1 P23458 1/20 0.42
TYK2 P29597 1/20 0.42
TAAR1 Q96RJ0 1/20 0.42
KMT2A Q03164 2/20 0.41
MEN1 O00255 1/20 0.41
CES2 O00748 1/20 0.41
CES1 P23141 1/20 0.41
ALDH1A1 P00352 1/20 0.40
LMNA P02545 1/20 0.40
PKM P14618 1/20 0.40
TLR7 Q9NYK1 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL3717023 0.98 BACE1 (0.49) BACE1GAAITGB2ICAM1ITGAL
SCHEMBL14333527 0.84 CES2 (0.50) BACE1ITGB2ICAM1ITGALKMT2A
Hydrochloric Acid SCHEMBL320643 0.82 CES2 (0.48) BACE1ITGB2ICAM1ITGALKMT2A
SCHEMBL22790324 0.81 GAA (0.47) BACE1GAAJAK2JAK1TYK2
SCHEMBL791513 0.81 GAA (0.47) BACE1GAAITGB2ICAM1ITGAL
SCHEMBL2867748 0.79 PBRM1 (0.58) GAAITGB2ICAM1ITGALPBRM1
Hydrochloric Acid SCHEMBL15568289 0.78 PBRM1 (0.56) GAAITGB2ICAM1ITGALPBRM1
Iodide SCHEMBL5204408 0.78 GAA (0.45) BACE1GAAJAK2JAK1TYK2
SCHEMBL1780411 0.77 TSHR (0.48) BACE1TAAR1KMT2AMEN1ALDH1A1
SCHEMBL7952512 0.77 CES2 (0.43) BACE1ITGB2ICAM1ITGALJAK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008084218-A1 BENZAZOLE DERIVATIVES FOR THE TREATMENT OF INFLAMMATIONS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2008-07-17 WO disclosed