SCHEMBL4737637

SCHEMBL4737637

CCOC(=O)[C@H](Cc1ccc(Nc2ncc(N)cc2N)cc1)NC1=CC(=O)C12CCCCC2

nearest known ligand 0.42

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ITGB1 P05556 5/20 0.42
ITGA4 P13612 5/20 0.42
ELANE P08246 1/20 0.33
NLRP3 Q96P20 1/20 0.32
XDH P47989 1/20 0.32
PPID Q08752 2/20 0.32
HTR1A P08908 1/20 0.31
HTR1D P28221 1/20 0.31
HTR2A P28223 1/20 0.31
HTR2C P28335 1/20 0.31
HTR7 P34969 1/20 0.31
HTR2B P41595 1/20 0.31
HTR5A P47898 1/20 0.31
HTR6 P50406 1/20 0.31
CPB2 Q96IY4 1/20 0.31
BACE1 P56817 1/20 0.30
ALDH1A1 P00352 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4735581 0.89 ITGB1 (0.46) ITGB1ITGA4ELANE
SCHEMBL4750224 0.85 ITGB1 (0.44) ITGB1ITGA4ELANENLRP3PPID
SCHEMBL4750220 0.85 ITGB1 (0.44) ITGB1ITGA4ELANENLRP3PPID
SCHEMBL4735983 0.84 ITGA4 (0.47) ITGB1ITGA4ELANE
SCHEMBL4736967 0.84 TDP1 (0.44) ITGB1ITGA4ALDH1A1
SCHEMBL4732361 0.83 KCNQ2 (0.39) ITGB1ITGA4PPID
SCHEMBL3832796 0.82 ITGB1 (0.47) ITGB1ITGA4ELANE
SCHEMBL3835880 0.81 ITGB1 (0.46) ITGB1ITGA4ELANENLRP3ALDH1A1
SCHEMBL4733784 0.80 MAPT (0.52) ITGB1ITGA4ALDH1A1
SCHEMBL4739188 0.79 ITGB1 (0.45) ITGB1ITGA4ELANE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008064830-A1 BICYCLIC AND HETEROBICYCLIC DERIVATIVES, PROCESSES FOR PREPARING THEM AND THEIR PHARMACEUTICAL USES UCB PHARMA, S.A. (BE) 2008-06-05 WO claimed
WO-2008064830-A1 BICYCLIC AND HETEROBICYCLIC DERIVATIVES, PROCESSES FOR PREPARING THEM AND THEIR PHARMACEUTICAL USES UCB PHARMA, S.A. (BE) 2008-06-05 WO disclosed