SCHEMBL4786839

SCHEMBL4786839

Cn1cc(-c2nc(N)nc3c2-c2cc(N)c(Cl)cc2CC3)cn1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PIKFYVE Q9Y2I7 2/20 0.39
TYMS P04818 1/20 0.39
ADORA2A P29274 1/20 0.36
AXL P30530 3/20 0.35
PGK1 P00558 1/20 0.35
CNR1 P21554 1/20 0.34
CNR2 P34972 1/20 0.34
IGF1R P08069 4/20 0.34
AURKA O14965 1/20 0.33
TTK P33981 1/20 0.33
AURKB Q96GD4 1/20 0.33
INCENP Q9NQS7 1/20 0.33
CSF1R P07333 1/20 0.33
CCNT1 O60563 2/20 0.33
CCNB2 O95067 2/20 0.33
CCNE2 O96020 2/20 0.33
CDK1 P06493 2/20 0.33
CCNB1 P14635 2/20 0.33
CCNE1 P24864 2/20 0.33
CDK2 P24941 2/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4736835 0.80 CCNT1 (0.40) CCNT1CCNB2CCNE2CDK1CCNB1
SCHEMBL4741246 0.80 TYMS (0.42) TYMSADORA2A
SCHEMBL4741259 0.79 TYMS (0.41) TYMSADORA2A
SCHEMBL4740440 0.78 TYMS (0.41) PIKFYVETYMSADORA2A
SCHEMBL4741224 0.77 HRH3 (0.53) TYMSADORA2A
SCHEMBL4737740 0.77 ADORA2A (0.46) TYMSADORA2A
SCHEMBL4739903 0.77 PIK3CA (0.41)
SCHEMBL14148428 0.76 TYMS (0.51) TYMS
SCHEMBL4741116 0.76 DHFR (0.40) TYMSADORA2A
SCHEMBL4741251 0.75 ADORA2A (0.43) TYMSADORA2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008086158-A1 BENZODIHYDROQUINAZOLINE AS PI3 KINASE INHIBITORS SMITHKLINE BEECHAM CORPORATION (US) 2008-07-17 WO disclosed