SCHEMBL4738145

SCHEMBL4738145

Cc1nc2c(OC(=O)C(C)(C)C)c(CC=C3Cc4ccccc4C3=O)c(C(=O)N(C)C)cc2n1C

nearest known ligand 0.35

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ACHE P22303 3/20 0.35
KMT2A Q03164 3/20 0.33
KDM4E B2RXH2 2/20 0.33
MEN1 O00255 2/20 0.33
BACE1 P56817 1/20 0.31
BCHE P06276 1/20 0.30
ALDH1A1 P00352 2/20 0.30
RAB9A P51151 2/20 0.30
SMN1; SMN2 Q16637 2/20 0.30
NPC1 O15118 1/20 0.30
S1PR4 O95977 1/20 0.30
GLA P06280 1/20 0.30
GAA P10253 1/20 0.30
HPGD P15428 1/20 0.30
S1PR1 P21453 1/20 0.30
MAOA P21397 1/20 0.30
MAOB P27338 1/20 0.30
MAPT P10636 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4738139 1.00 ACHE (0.35) ACHEKMT2AKDM4EMEN1BACE1
SCHEMBL4736286 0.83
SCHEMBL4734337 0.83 DUSP10 (0.31)
SCHEMBL4737851 0.83 CYP19A1 (0.32) ACHEKMT2AKDM4EMEN1BCHE
SCHEMBL4735621 0.82
SCHEMBL4735242 0.82 FNTA (0.31)
SCHEMBL4735017 0.82
SCHEMBL4739807 0.81 PTK2 (0.31)
SCHEMBL4735019 0.81 NQO2 (0.38) ACHEMAPT
SCHEMBL4739265 0.81

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008071765-A1 PHARMACEUTICALLY ACTIVE SPIRO-SUBSTITUTED BENZIMIDAZOLE DERIVATIVES NYCOMED GMBH (DE) 2008-06-19 WO disclosed