SCHEMBL4735019

SCHEMBL4735019

COc1ccc2c(c1)C(=CCc1c(C(=O)N(C)C)cc3c(nc(C)n3C)c1OC(=O)C(C)(C)C)CC2

nearest known ligand 0.38

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
NQO2 P16083 2/20 0.38
MTNR1A P48039 2/20 0.38
MTNR1B P49286 2/20 0.38
CYP19A1 P11511 5/20 0.32
CYP11B2 P19099 2/20 0.32
ACHE P22303 1/20 0.31
TP53 P04637 1/20 0.30
MAPT P10636 1/20 0.30
ABCB1 P08183 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4737851 0.94 CYP19A1 (0.32) NQO2MTNR1AMTNR1BCYP19A1CYP11B2
SCHEMBL4734337 0.92 DUSP10 (0.31)
SCHEMBL4738147 0.88 NQO2 (0.42) NQO2MTNR1AMTNR1BCYP19A1CYP11B2
SCHEMBL4736286 0.87
SCHEMBL4735017 0.86
SCHEMBL4735242 0.86 FNTA (0.31)
SCHEMBL4739807 0.85 PTK2 (0.31) CYP19A1CYP11B2
SCHEMBL4739210 0.81 MIF (0.36) NQO2MTNR1AMTNR1BCYP19A1CYP11B2
SCHEMBL4738139 0.81 ACHE (0.35) ACHEMAPT
SCHEMBL4738145 0.81 ACHE (0.35) ACHEMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008071765-A1 PHARMACEUTICALLY ACTIVE SPIRO-SUBSTITUTED BENZIMIDAZOLE DERIVATIVES NYCOMED GMBH (DE) 2008-06-19 WO disclosed