SCHEMBL4738510

SCHEMBL4738510

COC(=O)N1CCC(Nc2nc(Cl)nc(-c3cccc(F)c3)n2)CC1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
IDH1 O75874 2/20 0.42
IDH2 P48735 1/20 0.42
OPRM1 P35372 1/20 0.41
CCNT1 O60563 1/20 0.41
CSNK1E P49674 1/20 0.40
CYP1A2 P05177 1/20 0.39
CYP2D6 P10635 1/20 0.39
CYP2C19 P33261 1/20 0.39
MAPK14 Q16539 1/20 0.39
ACACB O00763 2/20 0.39
ACACA Q13085 2/20 0.39
RORC P51449 1/20 0.39
PDE4B Q07343 1/20 0.38
PDE4D Q08499 1/20 0.38
NOS1 P29475 1/20 0.38
NOS2 P35228 1/20 0.38
ALDH1A1 P00352 1/20 0.38
LMNA P02545 1/20 0.38
DNMT3A Q9Y6K1 1/20 0.38
CDK1 P06493 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4783578 0.88 CSNK1E (0.43) CSNK1EPDE4BPDE4DGRM5
SCHEMBL4784447 0.79 IDH1 (0.37) IDH1IDH2OPRM1CCNT1CSNK1E
SCHEMBL4784326 0.78 IDH1 (0.35) IDH1IDH2OPRM1MAPK14ACACB
SCHEMBL27172445 0.77 MAPK1 (0.49) IDH1ACACBACACARORCCDK1
SCHEMBL15102654 0.68 IDH1 (0.49) IDH1ALDH1A1
SCHEMBL29560753 0.68 IDH1 (0.49) IDH1ALDH1A1
SCHEMBL4998381 0.68 CDK2 (0.52) MAPK14NOS1NOS2LMNACDK1
SCHEMBL4786965 0.67 NT5E (0.46) ALDH1A1
SCHEMBL30414816 0.67 NT5E (0.46) ALDH1A1
SCHEMBL4785158 0.67 MAPK1 (0.35) CSNK1EPDE4BPDE4DGRM5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008072850-A1 TRIAZINE DERIVATIVES HAVING INHIBITORY ACTIVITY AGAINST ACETYL-COA CARBOXYLASE AMOREPACIFIC CORPORATION (KR) 2008-06-19 WO disclosed
WO-2008072850-A1 TRIAZINE DERIVATIVES HAVING INHIBITORY ACTIVITY AGAINST ACETYL-COA CARBOXYLASE AMOREPACIFIC CORPORATION (KR) 2008-06-19 WO disclosed