SCHEMBL4784447

SCHEMBL4784447

COC(=O)N1CCC(Nc2nc(-c3cccc(F)c3)nc(N3Cc4ccccc4C[C@@H]3CO)n2)CC1

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
IDH1 O75874 1/20 0.37
IDH2 P48735 1/20 0.37
ALDH1A1 P00352 2/20 0.36
MAPT P10636 2/20 0.36
DNMT3A Q9Y6K1 1/20 0.35
TP53 P04637 1/20 0.35
CDK1 P06493 1/20 0.35
CDK4 P11802 1/20 0.35
CCND1 P24385 1/20 0.35
CDK2 P24941 1/20 0.35
PTPN1 P18031 1/20 0.35
CCNT1 O60563 1/20 0.35
PDE4B Q07343 2/20 0.35
ACACB O00763 1/20 0.35
ACACA Q13085 1/20 0.35
OPRM1 P35372 1/20 0.34
HPGDS O60760 1/20 0.34
CHRM3 P20309 2/20 0.34
PDE4D Q08499 1/20 0.34
CSNK1E P49674 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4785161 0.91 CSNK1E (0.36) PDE4BPDE4DCSNK1E
SCHEMBL4785822 0.85 CTSL (0.40) ALDH1A1TP53PDE4BPDE4D
SCHEMBL4857757 0.84 DRD2 (0.44) ALDH1A1MAPT
SCHEMBL4784326 0.84 IDH1 (0.35) IDH1IDH2ALDH1A1DNMT3ATP53
SCHEMBL4738510 0.79 IDH1 (0.42) IDH1IDH2ALDH1A1DNMT3ACDK1
SCHEMBL4784054 0.76 PIK3CA (0.37) IDH1ALDH1A1TP53
SCHEMBL4784674 0.75 HRH4 (0.43) ALDH1A1TP53CDK2
SCHEMBL4785158 0.74 MAPK1 (0.35) TP53PDE4BPDE4DCSNK1E
SCHEMBL4782277 0.71 ADORA2A (0.35) ALDH1A1
SCHEMBL4785292 0.71 ROCK1 (0.35)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008072850-A1 TRIAZINE DERIVATIVES HAVING INHIBITORY ACTIVITY AGAINST ACETYL-COA CARBOXYLASE AMOREPACIFIC CORPORATION (KR) 2008-06-19 WO claimed
WO-2008072850-A1 TRIAZINE DERIVATIVES HAVING INHIBITORY ACTIVITY AGAINST ACETYL-COA CARBOXYLASE AMOREPACIFIC CORPORATION (KR) 2008-06-19 WO disclosed