SCHEMBL4739276

SCHEMBL4739276

Cc1c(F)cc(C(=O)Nc2ccnn2C)cc1-c1ccc(C(N)=O)cn1

nearest known ligand 0.46

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
MAPK14 Q16539 12/20 0.46
CYP2C9 P11712 7/20 0.46
MAPK11 Q15759 3/20 0.46
BUB1 O43683 1/20 0.45
PRKACG P22612 1/20 0.45
MAPKAPK2 P49137 1/20 0.45
ACSL5 Q9ULC5 1/20 0.45
STK24 Q9Y6E0 1/20 0.45
HPGDS O60760 2/20 0.43
LCK P06239 1/20 0.40
AKT1 P31749 1/20 0.38
NTRK1 P04629 1/20 0.37
KCNQ3 O43525 1/20 0.36
KCNQ2 O43526 1/20 0.36
MAPK8 P45983 1/20 0.35
MAPK10 P53779 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4800075 0.85 MAPK14 (0.65) MAPK14CYP2C9MAPK11BUB1PRKACG
SCHEMBL4738292 0.85 MAPK14 (0.65) MAPK14CYP2C9MAPK11BUB1PRKACG
SCHEMBL4680753 0.79 MAPK14 (0.46) MAPK14CYP2C9MAPK11BUB1PRKACG
SCHEMBL2214625 0.79 MAPK14 (0.40) MAPK14CYP2C9MAPK11BUB1PRKACG
SCHEMBL2216170 0.77 KDM4E (0.39) MAPK14CYP2C9MAPK11HPGDSNTRK1
SCHEMBL2213762 0.75 MAPK1 (0.44)
SCHEMBL2214850 0.75 MAPK14 (0.46) MAPK14HPGDSLCKKCNQ3KCNQ2
SCHEMBL14403123 0.75 P4HA1 (0.49) MAPK14CYP2C9MAPK11BUB1PRKACG
SCHEMBL14161063 0.74 MAPK14 (0.43) MAPK14HPGDSLCKKCNQ3KCNQ2
SCHEMBL4035180 0.74 MAPK14 (0.56) MAPK14HPGDSLCKKCNQ3KCNQ2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008071665-A1 A NICOTINAMIDE DERIVATIVE USEFUL AS P38 KINASE INHIBITOR SMITHKLINE BEECHAM CORPORATION (US) 2008-06-19 WO disclosed