SCHEMBL473975

SCHEMBL473975

COc1ccc(C(CO)C(c2cc(C)c(C#N)c(C)c2)C(F)(F)F)c(Cl)c1

nearest known ligand 0.33

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
S1PR1 P21453 1/20 0.33
S1PR3 Q99500 1/20 0.33
MAPT P10636 5/20 0.33
POLB P06746 2/20 0.33
TSHR P16473 2/20 0.33
CDK2 P24941 1/20 0.33
CLK1 P49759 1/20 0.33
NPSR1 Q6W5P4 1/20 0.33
MAPK1 P28482 1/20 0.33
KMT2A Q03164 3/20 0.32
RECQL P46063 1/20 0.32
KDM4E B2RXH2 6/20 0.32
ALDH1A1 P00352 5/20 0.32
GLA P06280 3/20 0.32
L3MBTL1 Q9Y468 3/20 0.32
TDP1 Q9NUW8 2/20 0.32
ABCC8 Q09428 1/20 0.32
KCNJ11 Q14654 1/20 0.32
NR3C1 P04150 1/20 0.32
PGR P06401 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL474058 0.86 ESR1 (0.34)
SCHEMBL473973 0.73 AR (0.41) S1PR1S1PR3MAPTPOLBTSHR
SCHEMBL473899 0.69 RECQL (0.42) S1PR1S1PR3POLBTSHRMAPK1
SCHEMBL3654236 0.69 LOXL2 (0.37) MAPTKMT2AKDM4EALDH1A1HPGD
SCHEMBL3658104 0.68 MRGPRX4 (0.42) KMT2AKDM4EALDH1A1HPGDMEN1
SCHEMBL3658899 0.68 NR1H4 (0.37) POLB
SCHEMBL3660073 0.63 MAPT (0.32) MAPTNPSR1ALDH1A1GAAHPGD
SCHEMBL474033 0.63 RECQL (0.45) MAPTPOLBTSHRMAPK1KMT2A
SCHEMBL3687105 0.62 SLC6A4 (0.44) MAPTCLK1KDM4EALDH1A1GLA
SCHEMBL13183805 0.61 KDM4E (0.37) MAPTPOLBMAPK1KMT2ARECQL

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2411365-A1 2,3-DIARYL- OR HETEROARYL-SUBSTITUTED 1,1,1-TRIFLUORO-2-HYDROXYPROPYL COMPOUNDS F. Hoffmann-La Roche AG (CH) 2012-02-01 EP disclosed
WO-2010108903-A1 2,3-DIARYL- OR HETEROARYL-SUBSTITUTED 1,1,1-TRIFLUORO-2-HYDROXYPROPYL COMPOUNDS F. HOFFMANN-LA ROCHE AG (CH) 2010-09-30 WO disclosed