SCHEMBL4739757

SCHEMBL4739757

COC(=O)c1ccc2ccc(Oc3ccnc([AsH]C(=O)OC(C)(C)C)c3)cc2c1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALOX15 P16050 2/20 0.39
HTT P42858 1/20 0.39
CYP19A1 P11511 1/20 0.38
CYP11B1 P15538 1/20 0.38
CYP11B2 P19099 1/20 0.38
CYP17A1 P05093 1/20 0.37
CYP3A4 P08684 1/20 0.37
HGFAC Q04756 1/20 0.36
PTPN11 Q06124 1/20 0.36
KDM4E B2RXH2 2/20 0.35
KDM6B O15054 1/20 0.35
KDM5C P41229 1/20 0.35
KDM4C Q9H3R0 1/20 0.35
KDM2A Q9Y2K7 1/20 0.35
KDM3A Q9Y4C1 1/20 0.35
ALDH1A1 P00352 1/20 0.35
HPGD P15428 1/20 0.35
NPSR1 Q6W5P4 1/20 0.35
NR1H4 Q96RI1 3/20 0.35
LCK P06239 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL546440 0.83 ALOX15 (0.41) ALOX15HTTCYP19A1CYP11B1CYP11B2
SCHEMBL546233 0.80 P2RX3 (0.45) ALOX15HTTCYP19A1CYP11B1CYP11B2
SCHEMBL545540 0.75 KDM4E (0.47) ALOX15HTTCYP19A1CYP11B1CYP11B2
Hydrochloric Acid SCHEMBL546682 0.74 KDM4E (0.46) ALOX15HTTCYP19A1CYP11B1CYP11B2
SCHEMBL19478119 0.73 BRAF (0.58) KDR
SCHEMBL545151 0.73 KDM4E (0.45) KDM4EKDM6BKDM5CKDM4CKDM2A
SCHEMBL545876 0.70 P2RX3 (0.46) KDM4ELCKDYRK1AKDR
SCHEMBL17598755 0.69 ELANE (0.58) ALOX15HTTCYP19A1CYP11B1CYP11B2
SCHEMBL27595732 0.69 KDM4E (0.58) KDM4EALDH1A1HPGDRAB9APLG
SCHEMBL545959 0.68 KDM4E (0.66) CYP11B1CYP11B2HGFACPTPN11KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1957460-A1 BICYCLIC COMPOUNDS WITH KINASE INHIBITORY ACTIVITY MILLENNIUM PHARMACEUTICALS, INC. (US) 2008-08-20 EP disclosed
WO-2007067444-A1 BICYCLIC COMPOUNDS WITH KINASE INHIBITORY ACTIVITY MILLENNIUM PHARMACEUTICALS, INC. (US) 2007-06-14 WO disclosed