SCHEMBL4740862

SCHEMBL4740862

CC1(C)CC(=O)C=C(Nc2c(N)ccnc2N)C1

nearest known ligand 0.58

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 9/20 0.58
L3MBTL1 Q9Y468 2/20 0.58
KDM4E B2RXH2 3/20 0.53
MEN1 O00255 2/20 0.51
TSHR P16473 2/20 0.51
KMT2A Q03164 2/20 0.51
GAA P10253 2/20 0.51
GLA P06280 1/20 0.51
MAPT P10636 1/20 0.51
ALOX15 P16050 1/20 0.51
CASP1 P29466 1/20 0.51
CASP7 P55210 1/20 0.51
HPGD P15428 2/20 0.46
PKM P14618 1/20 0.46
SMN1; SMN2 Q16637 2/20 0.45
TDP1 Q9NUW8 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13704104 0.81 KDM4E (0.59) ALDH1A1L3MBTL1KDM4EMEN1TSHR
SCHEMBL4743201 0.77 ALDH1A1 (0.50) ALDH1A1L3MBTL1KDM4EMEN1TSHR
SCHEMBL13704062 0.76 KDM4E (0.53) ALDH1A1L3MBTL1KDM4EMEN1TSHR
SCHEMBL14102109 0.76 KMT2A (0.63) ALDH1A1L3MBTL1KDM4EMEN1TSHR
SCHEMBL14106953 0.76 KDM4E (0.60) ALDH1A1L3MBTL1KDM4EMEN1TSHR
SCHEMBL28366538 0.73 ALDH1A1 (1.00) ALDH1A1L3MBTL1KDM4EMEN1TSHR
SCHEMBL13704047 0.73 ALDH1A1 (0.71) ALDH1A1L3MBTL1KDM4EMEN1TSHR
SCHEMBL4742790 0.70 KMT2A (0.54) ALDH1A1L3MBTL1KDM4EMEN1TSHR
SCHEMBL25791843 0.68 ALDH1A1 (0.73) ALDH1A1KDM4EMEN1TSHRKMT2A
SCHEMBL12821043 0.68 ALDH1A1 (0.61) ALDH1A1L3MBTL1KDM4EMEN1TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008099021-A1 DIBENZODIAZEPINONES USEFUL AS HEPATITIS C VIRUS INHIBITORS TIBOTEC PHARMACEUTICALS LTD. (IE) 2008-08-21 WO disclosed
WO-2008099021-A1 DIBENZODIAZEPINONES USEFUL AS HEPATITIS C VIRUS INHIBITORS TIBOTEC PHARMACEUTICALS LTD. (IE) 2008-08-21 WO disclosed