SCHEMBL4741268

SCHEMBL4741268

COc1ccc(-c2nc(N)nc3c2-c2cc(OC)ccc2CC3)cc1

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TYMS P04818 2/20 0.57
HRH3 Q9Y5N1 3/20 0.54
HRH2 P25021 2/20 0.54
MAPT P10636 3/20 0.49
KDM4E B2RXH2 2/20 0.49
ALDH1A1 P00352 2/20 0.49
MPI P34949 1/20 0.49
HTT P42858 2/20 0.47
ADORA1 P30542 3/20 0.46
KMT2A Q03164 1/20 0.46
ADORA2A P29274 3/20 0.44
NPY5R Q15761 1/20 0.43
TP53 P04637 1/20 0.43
TSHR P16473 1/20 0.43
MAPK1 P28482 1/20 0.43
MAPK10 P53779 1/20 0.43
PTK2B Q14289 1/20 0.43
NCOA1 Q15788 1/20 0.43
NCOA3 Q9Y6Q9 1/20 0.43
PDCD1 Q15116 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4741122 0.93 TYMS (0.55) TYMSHRH3HRH2MAPTKDM4E
SCHEMBL4739002 0.86 TYMS (0.51) TYMSHRH3HRH2MAPTKDM4E
SCHEMBL4741224 0.86 HRH3 (0.53) TYMSHRH3HRH2MAPTKDM4E
SCHEMBL4741223 0.82 TYMS (0.62) TYMSMAPTKDM4EALDH1A1MPI
SCHEMBL4741749 0.76 NPY5R (0.50) TYMSMAPTKDM4EALDH1A1MPI
SCHEMBL4740434 0.76 ADORA2A (0.51) TYMSHRH3HRH2MAPTKDM4E
SCHEMBL4787478 0.73 TYMS (0.49) TYMSMAPTKDM4EALDH1A1MPI
SCHEMBL6652286 0.72 TYMS (1.00) TYMS
SCHEMBL7000669 0.72 KDM4E (0.80) TYMSMAPTKDM4EALDH1A1MPI
Hydrochloric Acid SCHEMBL6844303 0.72 TYMS (0.98) TYMS

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008086158-A1 BENZODIHYDROQUINAZOLINE AS PI3 KINASE INHIBITORS SMITHKLINE BEECHAM CORPORATION (US) 2008-07-17 WO disclosed
WO-2008086158-A1 BENZODIHYDROQUINAZOLINE AS PI3 KINASE INHIBITORS SMITHKLINE BEECHAM CORPORATION (US) 2008-07-17 WO disclosed