SCHEMBL4741749

SCHEMBL4741749

CNc1nc2c(c(-c3ccccc3)n1)-c1cc(OC)ccc1CC2

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPY5R Q15761 2/20 0.50
ADORA1 P30542 6/20 0.48
ADORA2A P29274 4/20 0.48
TYMS P04818 1/20 0.47
ADORA2B P29275 1/20 0.46
KDM4E B2RXH2 3/20 0.42
L3MBTL1 Q9Y468 2/20 0.42
MAPK1 P28482 2/20 0.41
RECQL P46063 1/20 0.41
MAPT P10636 3/20 0.40
ALDH1A1 P00352 2/20 0.40
MPI P34949 1/20 0.40
IGF1R P08069 1/20 0.40
MAPK14 Q16539 1/20 0.40
HRH1 P35367 1/20 0.40
HRH4 Q9H3N8 1/20 0.40
MAOB P27338 1/20 0.40
TUBB4A P04350 1/20 0.39
TUBB P07437 1/20 0.39
TUBA3C P0DPH7 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4741122 0.84 TYMS (0.55) NPY5RADORA1ADORA2ATYMSADORA2B
SCHEMBL4741268 0.76 TYMS (0.57) NPY5RADORA1ADORA2ATYMSKDM4E
SCHEMBL4739002 0.69 TYMS (0.51) NPY5RADORA1ADORA2ATYMSKDM4E
SCHEMBL6835181 0.68 NPY5R (0.49) NPY5RTYMSKDM4EL3MBTL1MAPK1
SCHEMBL6835533 0.67 NPY5R (1.00) NPY5RTYMSKDM4EMAPTALDH1A1
SCHEMBL14148145 0.66 MAPT (0.50) ADORA1ADORA2ATYMSMAPTIGF1R
SCHEMBL4741223 0.66 TYMS (0.62) TYMSKDM4EMAPTALDH1A1MPI
SCHEMBL2340188 0.65 ALDH1A1 (0.62) NPY5RALDH1A1MAPK14LMNA
SCHEMBL6652286 0.64 TYMS (1.00) TYMS
SCHEMBL12567895 0.64 NPY5R (0.57) NPY5RKDM4EMAPTALDH1A1MPI

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008086158-A1 BENZODIHYDROQUINAZOLINE AS PI3 KINASE INHIBITORS SMITHKLINE BEECHAM CORPORATION (US) 2008-07-17 WO disclosed
WO-2008086158-A1 BENZODIHYDROQUINAZOLINE AS PI3 KINASE INHIBITORS SMITHKLINE BEECHAM CORPORATION (US) 2008-07-17 WO disclosed