SCHEMBL4741122

SCHEMBL4741122

COc1ccc2c(c1)-c1c(nc(N)nc1-c1ccccc1)CC2

nearest known ligand 0.55

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
TYMS P04818 1/20 0.55
NPY5R Q15761 2/20 0.52
ADORA2A P29274 9/20 0.47
ADORA1 P30542 7/20 0.47
KDM4E B2RXH2 3/20 0.47
ALDH1A1 P00352 2/20 0.47
MAPT P10636 2/20 0.47
MPI P34949 1/20 0.47
ADORA2B P29275 2/20 0.46
HRH2 P25021 1/20 0.46
HRH3 Q9Y5N1 1/20 0.46
HTT P42858 1/20 0.45
ACHE P22303 2/20 0.44
MAOB P27338 1/20 0.44
L3MBTL1 Q9Y468 2/20 0.43
MAPK1 P28482 1/20 0.43
RECQL P46063 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4741268 0.93 TYMS (0.57) TYMSNPY5RADORA2AADORA1KDM4E
SCHEMBL4739002 0.84 TYMS (0.51) TYMSNPY5RADORA2AADORA1KDM4E
SCHEMBL4741749 0.84 NPY5R (0.50) TYMSNPY5RADORA2AADORA1KDM4E
SCHEMBL4741223 0.80 TYMS (0.62) TYMSKDM4EALDH1A1MAPTMPI
SCHEMBL4741224 0.79 HRH3 (0.53) TYMSADORA2AADORA1KDM4EALDH1A1
SCHEMBL4740434 0.79 ADORA2A (0.51) TYMSADORA2AADORA1KDM4EALDH1A1
SCHEMBL8067781 0.77 ACHE (0.65) NPY5RADORA2AADORA1KDM4EADORA2B
SCHEMBL4741246 0.77 TYMS (0.42) TYMSADORA2AADORA1KDM4EALDH1A1
SCHEMBL4739911 0.74 TYMS (0.52) TYMSADORA2AADORA1ADORA2BACHE
SCHEMBL8072372 0.74 ADORA2A (0.73) ADORA2AADORA1ADORA2BHRH3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008086158-A1 BENZODIHYDROQUINAZOLINE AS PI3 KINASE INHIBITORS SMITHKLINE BEECHAM CORPORATION (US) 2008-07-17 WO disclosed
WO-2008086158-A1 BENZODIHYDROQUINAZOLINE AS PI3 KINASE INHIBITORS SMITHKLINE BEECHAM CORPORATION (US) 2008-07-17 WO disclosed