SCHEMBL4787478

SCHEMBL4787478

COc1ccc2c(c1)-c1c(nc(N)nc1Nc1cc(OC)c(OC)c(OC)c1)CC2

nearest known ligand 0.49

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
TYMS P04818 1/20 0.49
BRAF P15056 6/20 0.48
EGFR P00533 2/20 0.43
LCK P06239 2/20 0.43
MAPT P10636 2/20 0.41
TP53 P04637 1/20 0.41
DHFR P00374 1/20 0.40
KDM4E B2RXH2 1/20 0.40
ALDH1A1 P00352 1/20 0.40
MPI P34949 1/20 0.40
MEN1 O00255 1/20 0.39
KMT2A Q03164 1/20 0.39
GAK O14976 2/20 0.39
RIPK2 O43353 2/20 0.39
COQ8A Q8NI60 2/20 0.39
NLK Q9UBE8 2/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4741223 0.75 TYMS (0.62) TYMSMAPTTP53DHFRKDM4E
SCHEMBL4737442 0.74 MAPT (0.41) BRAFMAPTKDM4EALDH1A1MEN1
SCHEMBL4741268 0.73 TYMS (0.57) TYMSMAPTTP53DHFRKDM4E
SCHEMBL4741122 0.71 TYMS (0.55) TYMSMAPTKDM4EALDH1A1MPI
SCHEMBL7237418 0.71 FYN (0.65) BRAFLCKMAPTTP53KDM4E
SCHEMBL4739002 0.70 TYMS (0.51) TYMSMAPTKDM4EALDH1A1MPI
SCHEMBL12391883 0.67 HIF1A (0.54) EGFRMEN1KMT2A
SCHEMBL6652286 0.66 TYMS (1.00) TYMS
SCHEMBL6997904 0.66 FYN (0.61) BRAFLCKMAPTTP53KDM4E
Hydrochloric Acid SCHEMBL6844303 0.65 TYMS (0.98) TYMS

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008086158-A1 BENZODIHYDROQUINAZOLINE AS PI3 KINASE INHIBITORS SMITHKLINE BEECHAM CORPORATION (US) 2008-07-17 WO disclosed
WO-2008086158-A1 BENZODIHYDROQUINAZOLINE AS PI3 KINASE INHIBITORS SMITHKLINE BEECHAM CORPORATION (US) 2008-07-17 WO disclosed