SCHEMBL4741648

SCHEMBL4741648

O=CCC(CC(=O)OC(=O)C(F)(F)F)NC(=O)c1cnc2cc(C(F)(F)F)ccc2c1N1CCCCC1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
THRB P10828 1/20 0.43
MAPT P10636 3/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
ALDH1A1 P00352 1/20 0.33
CCNC P24863 1/20 0.33
CDK8 P49336 1/20 0.33
KDR P35968 1/20 0.32
SRPK2 P78362 1/20 0.32
SRPK1 Q96SB4 1/20 0.32
SRPK3 Q9UPE1 1/20 0.32
MMP1 P03956 1/20 0.32
MMP9 P14780 1/20 0.32
MMP13 P45452 1/20 0.32
CTNNB1 P35222 1/20 0.32
TCF7L2 Q9NQB0 1/20 0.32
MEN1 O00255 2/20 0.32
KMT2A Q03164 2/20 0.32
PDE2A O00408 1/20 0.32
KDM4E B2RXH2 1/20 0.32
MCHR1 Q99705 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4739980 0.86 THRB (0.44) THRBMAPTSMN1; SMN2ALDH1A1CCNC
SCHEMBL4785503 0.79 THRB (0.45) THRBMAPTSMN1; SMN2ALDH1A1CASP3
SCHEMBL4742145 0.79 THRB (0.43) THRBMMP1MMP9MMP13PDGFRB
SCHEMBL4742120 0.79 THRB (0.43) THRBMMP1MMP9MMP13PDGFRB
SCHEMBL4741630 0.75 THRB (0.46) THRBMAPTSMN1; SMN2CCNCCDK8
SCHEMBL4742128 0.74 THRB (0.45) THRBMAPTSMN1; SMN2CCNCCDK8
SCHEMBL4743041 0.73 THRB (0.55) THRBMAPTSMN1; SMN2ALDH1A1CCNC
SCHEMBL4742554 0.69 TP53 (0.36) MAPTSMN1; SMN2ALDH1A1MEN1KMT2A
Trifluoroacetic Acid SCHEMBL4742140 0.68 THRB (0.43) THRBSMN1; SMN2ALDH1A1MMP1MMP9
Trifluoroacetic Acid SCHEMBL4785493 0.68 THRB (0.45) THRBMAPTSMN1; SMN2ALDH1A1MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008093940-A1 QUINOLINE DERIVATIVES AS CASPASE-3 INHIBITOR, PREPARATION PROCESS FOR THE SAME AND PHARMACEUTICAL COMPOSITION COMPRISING THE SAME YUNGJIN PHARMACEUTICAL CO., LTD. (KR) 2008-08-07 WO disclosed