SCHEMBL4741630

SCHEMBL4741630

CC(C)(C)OC(=O)CC(NC(=O)c1cnc2cc(C(F)(F)F)ccc2c1N1CCCCC1)C(=O)CF

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
THRB P10828 1/20 0.46
CYP8B1 Q9UNU6 6/20 0.36
CASP3 P42574 1/20 0.36
CASP6 P55212 1/20 0.36
CASP8 Q14790 1/20 0.36
MAPT P10636 2/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
CCNC P24863 1/20 0.35
CDK8 P49336 1/20 0.35
KDR P35968 2/20 0.35
TEK Q02763 1/20 0.35
SRPK2 P78362 1/20 0.35
SRPK1 Q96SB4 1/20 0.35
SRPK3 Q9UPE1 1/20 0.35
PDE2A O00408 1/20 0.34
MMP1 P03956 1/20 0.34
MMP9 P14780 1/20 0.34
MMP13 P45452 1/20 0.34
CYP3A4 P08684 1/20 0.34
UGCG Q16739 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4785468 0.92 THRB (0.45) THRBCYP8B1MMP1MMP9MMP13
SCHEMBL4743062 0.92 THRB (0.47) THRBCASP3CASP6CASP8MAPT
SCHEMBL4739980 0.89 THRB (0.44) THRBCYP8B1CASP3CASP6CASP8
SCHEMBL4742128 0.88 THRB (0.45) THRBCYP8B1MAPTSMN1; SMN2CCNC
SCHEMBL4742120 0.81 THRB (0.43) THRBCYP8B1CASP3MMP1MMP9
SCHEMBL4742145 0.81 THRB (0.43) THRBCYP8B1MMP1MMP9MMP13
SCHEMBL4785503 0.81 THRB (0.45) THRBCASP3CASP6CASP8MAPT
SCHEMBL4785519 0.80 THRB (0.44) THRBCYP8B1MMP1MMP9MMP13
SCHEMBL4743466 0.80 THRB (0.46) THRBMAPTSMN1; SMN2
SCHEMBL4739339 0.80 MET (0.46) THRBMAPTSMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008093940-A1 QUINOLINE DERIVATIVES AS CASPASE-3 INHIBITOR, PREPARATION PROCESS FOR THE SAME AND PHARMACEUTICAL COMPOSITION COMPRISING THE SAME YUNGJIN PHARMACEUTICAL CO., LTD. (KR) 2008-08-07 WO disclosed