SCHEMBL4743041

SCHEMBL4743041

O=C(O)c1cnc2cc(C(F)(F)F)ccc2c1N1CCCCC1

nearest known ligand 0.55

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
THRB P10828 1/20 0.55
MAPT P10636 1/20 0.43
SMN1; SMN2 Q16637 1/20 0.43
ALDH1A1 P00352 2/20 0.43
CYP8B1 Q9UNU6 3/20 0.43
CCNC P24863 1/20 0.42
CDK8 P49336 1/20 0.42
ADRB2 P07550 1/20 0.41
NCF1 P14598 1/20 0.41
LIPG Q9Y5X9 1/20 0.40
KDR P35968 1/20 0.40
SRPK2 P78362 1/20 0.40
SRPK1 Q96SB4 1/20 0.40
SRPK3 Q9UPE1 1/20 0.40
CSF1R P07333 1/20 0.39
KDM4E B2RXH2 1/20 0.39
HPGD P15428 1/20 0.39
HSD17B10 Q99714 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4743063 0.88 THRB (0.56) THRBMAPTSMN1; SMN2ALDH1A1HSD17B10
SCHEMBL4743443 0.88 THRB (0.53) THRBSMN1; SMN2ALDH1A1CYP8B1ADRB2
SCHEMBL4739993 0.82 THRB (0.54) THRBMAPTSMN1; SMN2CYP8B1HPGD
SCHEMBL3887756 0.77 ALDH1A1 (0.46) THRBALDH1A1KDRCSF1RKDM4E
SCHEMBL30592902 0.77 ALDH1A1 (0.46) THRBALDH1A1KDRCSF1RKDM4E
Hydrochloric Acid SCHEMBL11870232 0.76 ALDH1A1 (0.45) THRBALDH1A1KDRCSF1RKDM4E
SCHEMBL438818 0.76 ALDH1A1 (0.53) THRBALDH1A1KDRCSF1RKDM4E
SCHEMBL4466003 0.76 SORT1 (0.46) THRBALDH1A1KDRCSF1RKDM4E
SCHEMBL1644467 0.76 THRB (0.46) THRBALDH1A1KDRCSF1RKDM4E
SCHEMBL4741630 0.74 THRB (0.46) THRBMAPTSMN1; SMN2CYP8B1CCNC

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008093940-A1 QUINOLINE DERIVATIVES AS CASPASE-3 INHIBITOR, PREPARATION PROCESS FOR THE SAME AND PHARMACEUTICAL COMPOSITION COMPRISING THE SAME YUNGJIN PHARMACEUTICAL CO., LTD. (KR) 2008-08-07 WO disclosed