SCHEMBL4742147

SCHEMBL4742147

CC(C)(C)OC(=O)N1CCN(c2c(C(=O)O)cnc3c([N+](=O)[O-])cccc23)CC1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LMNA P02545 4/20 0.48
MAPT P10636 4/20 0.48
ALDH1A1 P00352 3/20 0.48
MET P08581 2/20 0.48
CKS1B P61024 2/20 0.44
SKP1 P63208 2/20 0.44
SKP2 Q13309 2/20 0.44
PTPN11 Q06124 1/20 0.44
SMN1; SMN2 Q16637 2/20 0.42
HTT P42858 2/20 0.42
MITF O75030 1/20 0.42
GBA1 P04062 2/20 0.41
KCNH2 Q12809 1/20 0.41
KIT P10721 1/20 0.40
MTOR P42345 1/20 0.40
RAB9A P51151 1/20 0.40
SIRT2 Q8IXJ6 1/20 0.40
ACHE P22303 1/20 0.40
POLB P06746 1/20 0.40
KDM4E B2RXH2 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4742099 0.88 LMNA (0.55) LMNAMAPTALDH1A1SMN1; SMN2HTT
SCHEMBL4743456 0.85 MAPT (0.47) MAPTCKS1BSKP1SKP2PTPN11
SCHEMBL4743444 0.84 USP2 (0.54) LMNAMAPTCKS1BSKP1SKP2
SCHEMBL31220479 0.84 ALDH1A1 (0.56) LMNAMAPTALDH1A1METCKS1B
SCHEMBL2977592 0.81 ALDH1A1 (0.63) LMNAMAPTALDH1A1METCKS1B
SCHEMBL4743406 0.80 MET (0.39) LMNAMAPTALDH1A1METCKS1B
SCHEMBL4742143 0.80 ALDH1A1 (0.58) LMNAMAPTALDH1A1METCKS1B
SCHEMBL4786909 0.80 MET (0.39) LMNAMAPTALDH1A1METPTPN11
SCHEMBL28520810 0.78 MTOR (0.64) LMNAMAPTALDH1A1SMN1; SMN2HTT
SCHEMBL2973720 0.76 ALDH1A1 (0.73) LMNAMAPTALDH1A1METSMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008093940-A1 QUINOLINE DERIVATIVES AS CASPASE-3 INHIBITOR, PREPARATION PROCESS FOR THE SAME AND PHARMACEUTICAL COMPOSITION COMPRISING THE SAME YUNGJIN PHARMACEUTICAL CO., LTD. (KR) 2008-08-07 WO disclosed