SCHEMBL4742591

SCHEMBL4742591

CCOC(=O)c1cnc2cc(C(F)(F)F)ccc2c1N1CCN(C(=O)OC(C)(C)C)CC1

nearest known ligand 0.72

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
THRB P10828 1/20 0.72
MEN1 O00255 5/20 0.53
KMT2A Q03164 5/20 0.53
HPGD P15428 1/20 0.50
SMN1; SMN2 Q16637 1/20 0.50
MAPK10 P53779 1/20 0.49
MAPT P10636 3/20 0.49
ALDH1A1 P00352 3/20 0.49
NPSR1 Q6W5P4 2/20 0.47
USP2 O75604 1/20 0.47
TP53 P04637 1/20 0.47
MAPK1 P28482 1/20 0.47
RECQL P46063 1/20 0.47
HSD17B10 Q99714 1/20 0.47
GAA P10253 1/20 0.47
PDGFRB P09619 2/20 0.46
LMNA P02545 1/20 0.46
PDE6D O43924 1/20 0.46
PDE5A O76074 1/20 0.46
PDE6A P16499 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4742620 0.89 THRB (0.64) THRBMEN1KMT2AMAPK10MAPT
SCHEMBL4739993 0.88 THRB (0.54) THRBHPGDSMN1; SMN2MAPTPDGFRB
SCHEMBL4742104 0.84 MAPT (0.53) THRBMEN1KMT2ASMN1; SMN2MAPK10
SCHEMBL4742585 0.84 THRB (0.75) THRBMEN1KMT2AMAPK10MAPT
SCHEMBL4743046 0.84 THRB (0.78) THRBMEN1KMT2ASMN1; SMN2MAPK10
SCHEMBL22396176 0.84 MAPT (0.59) THRBMEN1KMT2AMAPK10MAPT
SCHEMBL2943134 0.83 PDGFRB (0.63) THRBMEN1KMT2ASMN1; SMN2MAPK10
SCHEMBL25656123 0.82 MEN1 (0.55) THRBMEN1KMT2AMAPK10MAPT
SCHEMBL4785451 0.81 MAPK1 (0.72) MEN1KMT2ASMN1; SMN2MAPTALDH1A1
SCHEMBL23726472 0.80 PDGFRB (0.59) THRBMEN1KMT2ASMN1; SMN2MAPK10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008093940-A1 QUINOLINE DERIVATIVES AS CASPASE-3 INHIBITOR, PREPARATION PROCESS FOR THE SAME AND PHARMACEUTICAL COMPOSITION COMPRISING THE SAME YUNGJIN PHARMACEUTICAL CO., LTD. (KR) 2008-08-07 WO disclosed