SCHEMBL4742620

SCHEMBL4742620

CCOC(=O)c1cnc2cc(F)ccc2c1N1CCN(C(=O)OC(C)(C)C)CC1

nearest known ligand 0.64

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
THRB P10828 1/20 0.64
MEN1 O00255 4/20 0.57
KMT2A Q03164 4/20 0.57
MAPT P10636 5/20 0.52
MAPK10 P53779 1/20 0.51
ALDH1A1 P00352 2/20 0.50
NPSR1 Q6W5P4 3/20 0.49
LMNA P02545 2/20 0.49
GAA P10253 1/20 0.49
CYP8B1 Q9UNU6 1/20 0.48
PDGFRB P09619 1/20 0.47
KDM4E B2RXH2 1/20 0.47
GLA P06280 1/20 0.47
HTT P42858 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22396176 0.93 MAPT (0.59) THRBMEN1KMT2AMAPTMAPK10
SCHEMBL4742591 0.89 THRB (0.72) THRBMEN1KMT2AMAPTMAPK10
SCHEMBL4743436 0.88 SMN1; SMN2 (0.48) THRBMAPTALDH1A1LMNA
SCHEMBL4742104 0.86 MAPT (0.53) THRBMEN1KMT2AMAPTMAPK10
SCHEMBL2943134 0.84 PDGFRB (0.63) THRBMEN1KMT2AMAPTMAPK10
SCHEMBL25656123 0.83 MEN1 (0.55) THRBMEN1KMT2AMAPTMAPK10
SCHEMBL4741642 0.81 MAPT (0.64) MEN1KMT2AMAPTALDH1A1NPSR1
SCHEMBL23726472 0.81 PDGFRB (0.59) THRBMEN1KMT2AMAPTMAPK10
SCHEMBL30080115 0.81 PDGFRB (0.59) THRBMEN1KMT2AMAPTMAPK10
SCHEMBL22395760 0.80 ALDH1A1 (0.52) ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008093940-A1 QUINOLINE DERIVATIVES AS CASPASE-3 INHIBITOR, PREPARATION PROCESS FOR THE SAME AND PHARMACEUTICAL COMPOSITION COMPRISING THE SAME YUNGJIN PHARMACEUTICAL CO., LTD. (KR) 2008-08-07 WO disclosed