SCHEMBL4743218

SCHEMBL4743218

C[C@@H](c1ccccc1I)[N@@]1CC1(I)CO

nearest known ligand 0.32

Predicted protein targets (top 1)

geneUniProtsupporting neighboursconfidence
TSHR P16473 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4726066 0.80 CYP2D6 (0.43)
SCHEMBL4725612 0.68 TSHR (0.33) TSHR
SCHEMBL25009948 0.65 TSHR (0.42) TSHR
SCHEMBL3923412 0.64 KCNA3 (0.38)
SCHEMBL6682974 0.63 TSHR (0.59) TSHR
SCHEMBL23205864 0.63 TSHR (0.59) TSHR
SCHEMBL27458230 0.63 TSHR (0.59) TSHR
SCHEMBL25167464 0.63 KDM4E (0.33) TSHR
SCHEMBL4419612 0.62 GABRA1 (0.41) TSHR
SCHEMBL535657 0.62 GABRA1 (0.41) TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008109286-A1 METHODS FOR TREATING COGNITIVE DISORDERS USING 1-ARYL-1-HYDROXY-2,3-DIAMINO-PROPYL AMINES, 1-HETEROARYL-1-HYDROXY-2,3-DIAMINO-PROPYL AMINES AND RELATED COMPOUNDS ALLERGAN, INC. (US) 2008-09-12 WO disclosed
WO-2008109287-A1 METHODS FOR TREATING COGNITIVE DISORDERS USING 1-BENZYL-1-HYDROXY-2,3-DIAMINO-PROPYL AMINES, 3-BENZYL-3-HYDROXY-2-AMINO-PROPIONIC ACID AMIDES AND RELATED COMPOUNDS ALLERGAN, INC. (US) 2008-09-12 WO disclosed