SCHEMBL4726066

SCHEMBL4726066

C[C@@H](c1ccccc1)[N@@]1CC1(I)CO

nearest known ligand 0.43

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
CYP2D6 P10635 2/20 0.43
OPRM1 P35372 2/20 0.40
OPRD1 P41143 2/20 0.40
OPRK1 P41145 2/20 0.40
OPRL1 P41146 2/20 0.40
MC4R P32245 1/20 0.39
ALDH1A1 P00352 2/20 0.36
TRPA1 O75762 4/20 0.36
HPGD P15428 2/20 0.36
MEN1 O00255 1/20 0.35
KMT2A Q03164 1/20 0.35
HSD17B10 Q99714 1/20 0.35
HSD11B1 P28845 1/20 0.35
CYP1A2 P05177 1/20 0.34
HIF1A Q16665 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4743218 0.80 TSHR (0.32)
SCHEMBL10568119 0.72 CYP2D6 (0.55) CYP2D6OPRM1OPRD1OPRK1OPRL1
SCHEMBL4728306 0.70 CYP2D6 (0.43) CYP2D6OPRM1OPRD1OPRK1OPRL1
SCHEMBL7089368 0.68 ALDH1A1 (0.39) CYP2D6OPRM1OPRD1OPRK1OPRL1
SCHEMBL9683895 0.66 CYP2D6 (0.55) CYP2D6OPRM1OPRD1OPRK1OPRL1
SCHEMBL84798 0.66 CYP2D6 (0.46) CYP2D6OPRM1OPRD1OPRK1OPRL1
SCHEMBL85400 0.66 CYP2D6 (0.46) CYP2D6OPRM1OPRD1OPRK1OPRL1
SCHEMBL2337932 0.65 CYP2D6 (0.65) CYP2D6OPRM1OPRD1OPRK1OPRL1
SCHEMBL4922997 0.65 LMNA (0.55) CYP2D6OPRM1OPRD1OPRK1OPRL1
SCHEMBL7291562 0.65 LMNA (0.55) CYP2D6OPRM1OPRD1OPRK1OPRL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008109287-A1 METHODS FOR TREATING COGNITIVE DISORDERS USING 1-BENZYL-1-HYDROXY-2,3-DIAMINO-PROPYL AMINES, 3-BENZYL-3-HYDROXY-2-AMINO-PROPIONIC ACID AMIDES AND RELATED COMPOUNDS ALLERGAN, INC. (US) 2008-09-12 WO disclosed
WO-2008011487-A2 L-BENZYL-L-HYDR0XY-2, 3-DIAMIN0-PROPYL AMINES AND 3-BENZYL-3-HYDROXY-2-AMINO-PROPIONICACID AMIDES FOR CHRONIC PAIN ALLERGAN, INC. (US) 2008-01-24 WO disclosed