SCHEMBL4743436

SCHEMBL4743436

CC(C)(C)OC(=O)N1CCN(c2c(C(=O)O)cnc3cc(F)ccc23)CC1

nearest known ligand 0.48

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 1/20 0.48
THRB P10828 2/20 0.47
CKS1B P61024 1/20 0.44
SKP1 P63208 1/20 0.44
SKP2 Q13309 1/20 0.44
PTPN11 Q06124 1/20 0.43
ALDH1A1 P00352 7/20 0.43
LMNA P02545 2/20 0.43
KIT P10721 1/20 0.42
CCNC P24863 1/20 0.42
CDK8 P49336 1/20 0.42
GPR119 Q8TDV5 2/20 0.42
GRIA1 P42261 1/20 0.41
TP53 P04637 1/20 0.41
MAPT P10636 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22395760 0.92 ALDH1A1 (0.52) SMN1; SMN2ALDH1A1CCNCCDK8
SCHEMBL4739993 0.88 THRB (0.54) SMN1; SMN2THRBCKS1BSKP1SKP2
SCHEMBL4742620 0.88 THRB (0.64) THRBALDH1A1LMNAMAPT
SCHEMBL4742143 0.84 ALDH1A1 (0.58) SMN1; SMN2CKS1BSKP1SKP2PTPN11
SCHEMBL4785479 0.80 THRB (0.42) SMN1; SMN2THRBCKS1BSKP1SKP2
SCHEMBL22396176 0.80 MAPT (0.59) THRBALDH1A1LMNATP53MAPT
SCHEMBL4743456 0.80 MAPT (0.47) SMN1; SMN2THRBCKS1BSKP1SKP2
SCHEMBL23727334 0.79 MAPT (0.52) SMN1; SMN2CKS1BSKP1SKP2ALDH1A1
SCHEMBL30080180 0.79 MAPT (0.52) SMN1; SMN2CKS1BSKP1SKP2ALDH1A1
SCHEMBL30080182 0.79 MAPT (0.52) SMN1; SMN2CKS1BSKP1SKP2ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008093940-A1 QUINOLINE DERIVATIVES AS CASPASE-3 INHIBITOR, PREPARATION PROCESS FOR THE SAME AND PHARMACEUTICAL COMPOSITION COMPRISING THE SAME YUNGJIN PHARMACEUTICAL CO., LTD. (KR) 2008-08-07 WO disclosed