SCHEMBL4743517

SCHEMBL4743517

NCC(c1ccccc1)c1cc(C(F)(F)F)cc(C(F)(F)F)c1

nearest known ligand 0.59

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 2/20 0.59
TAAR1 Q96RJ0 1/20 0.59
IDO1 P14902 2/20 0.56
TDO2 P48775 2/20 0.56
PNMT P11086 1/20 0.53
TACR1 P25103 13/20 0.51
CACNA1F O60840 1/20 0.50
CACNA1D Q01668 1/20 0.50
CACNA1S Q13698 1/20 0.50
CACNA1C Q13936 1/20 0.50
CHRNB2 P17787 1/20 0.50
CHRNA4 P43681 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL605443 0.85 HTR2A (0.64) HTR2ATAAR1PNMTCACNA1CCHRNB2
SCHEMBL7412490 0.78 TACR1 (0.46) IDO1TDO2PNMTTACR1CACNA1F
2,2,2-Trifluoroethanaminium SCHEMBL4716808 0.78 HTR2A (0.73) HTR2ATAAR1PNMTCHRNB2CHRNA4
SCHEMBL149259 0.77 HTR2A (1.00) HTR2ATAAR1CHRNB2CHRNA4
SCHEMBL3914167 0.76 PNMT (0.59) HTR2ATAAR1IDO1TDO2PNMT
SCHEMBL19668650 0.75 SLC6A4 (0.58) HTR2AIDO1TDO2TACR1CACNA1F
Bromide SCHEMBL6737914 0.75 HTR2A (0.94) HTR2ATAAR1CHRNB2CHRNA4
Water SCHEMBL28365853 0.75 HTR2A (0.94) HTR2ATAAR1CHRNB2CHRNA4
Hydrochloric Acid SCHEMBL8550503 0.75 HTR2A (0.94) HTR2ATAAR1CHRNB2CHRNA4
SCHEMBL1581317 0.74 PNMT (0.45) HTR2ATAAR1PNMTCACNA1CCHRNB2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008106633-A1 METHODS OF USING BENZODIOXINE COMPOUNDS IN TREATING SODIUM CHANNEL-MEDIATED DISEASES OR CONDITIONS XENON PHARMACEUTICALS INC. (CA) 2008-09-04 WO disclosed