SCHEMBL7412490

SCHEMBL7412490

COc1ccccc1C(CN)c1cc(C(F)(F)F)cc(C(F)(F)F)c1

nearest known ligand 0.46

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
TACR1 P25103 10/20 0.46
IDO1 P14902 3/20 0.46
TDO2 P48775 3/20 0.46
CTSA P10619 2/20 0.42
CACNA1F O60840 1/20 0.42
CACNA1D Q01668 1/20 0.42
CACNA1S Q13698 1/20 0.42
CACNA1C Q13936 1/20 0.42
PNMT P11086 1/20 0.40
AKR1C3 P42330 1/20 0.40
AKR1C2 P52895 1/20 0.40
TACR3 P29371 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7409508 0.89 PNMT (0.51) TACR1IDO1TDO2PNMTAKR1C3
SCHEMBL21495213 0.80 IDO1 (0.56) IDO1TDO2
SCHEMBL2086020 0.80 IDO1 (0.56) IDO1TDO2
SCHEMBL4743517 0.78 HTR2A (0.59) TACR1IDO1TDO2CACNA1FCACNA1D
SCHEMBL14387383 0.71 SLC6A2 (0.48) IDO1TDO2CACNA1C
SCHEMBL7422189 0.70 KMT2A (0.43) IDO1TDO2CACNA1C
SCHEMBL6001132 0.68 TAAR1 (0.50) IDO1TDO2
SCHEMBL6993305 0.67 ADRA2A (0.40)
SCHEMBL6001484 0.67 HRH1 (0.59) IDO1TDO2
SCHEMBL17529671 0.67 CA1 (0.50) IDO1TDO2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1988003147-A1 SELECTED N6-SUBSTITUTED ADENOSINES HAVING SELECTIVE A2 BINDING ACTIVITY WARNER-LAMBERT COMPANY (US) 1988-05-05 WO disclosed