SCHEMBL4743568

SCHEMBL4743568

O=C1CSC(c2cccc(C(F)(F)F)c2)N1c1ccc(Oc2ccc(Cl)c(Cl)c2)cc1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 2/20 0.53
ALDH1A1 P00352 3/20 0.49
HTT P42858 1/20 0.49
NPSR1 Q6W5P4 1/20 0.49
HTR7 P34969 2/20 0.48
GFER P55789 4/20 0.47
CA1 P00915 3/20 0.47
CA2 P00918 3/20 0.47
CA9 Q16790 3/20 0.47
CYP1A2 P05177 1/20 0.46
GAA P10253 1/20 0.46
CYP2C9 P11712 1/20 0.46
CYP2C19 P33261 1/20 0.46
SMN1; SMN2 Q16637 1/20 0.46
CACNA1B Q00975 1/20 0.46
MEN1 O00255 1/20 0.43
TUBB4A P04350 1/20 0.42
TUBB P07437 1/20 0.42
TUBA3C P0DPH7 1/20 0.42
TUBA1B P68363 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4744303 0.94 HTR7 (0.48) KMT2AALDH1A1HTTNPSR1HTR7
SCHEMBL4743511 0.91 KMT2A (0.55) KMT2AALDH1A1HTTNPSR1HTR7
SCHEMBL4747346 0.89 KMT2A (0.53) KMT2AALDH1A1HTTNPSR1HTR7
SCHEMBL4743939 0.89 ALDH1A1 (0.61) KMT2AALDH1A1HTTNPSR1HTR7
SCHEMBL4746786 0.88 KMT2A (0.62) KMT2AALDH1A1HTTNPSR1HTR7
SCHEMBL14069571 0.88 KMT2A (0.56) KMT2AALDH1A1HTTNPSR1HTR7
SCHEMBL4744248 0.87 HTR7 (0.49) KMT2AALDH1A1HTTNPSR1HTR7
SCHEMBL4744239 0.87 KMT2A (0.64) KMT2AALDH1A1HTTNPSR1HTR7
SCHEMBL4743988 0.87 GFER (0.57) KMT2AALDH1A1HTTNPSR1HTR7
SCHEMBL4743915 0.87 KMT2A (0.55) KMT2AALDH1A1HTTNPSR1HTR7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008112674-A1 COMPOUNDS AND COMPOSITIONS AS INHIBITORS OF CANNABINOID RECEPTOR 1 ACTIVITY IRM LLC (BM) 2008-09-18 WO claimed
WO-2008112674-A1 COMPOUNDS AND COMPOSITIONS AS INHIBITORS OF CANNABINOID RECEPTOR 1 ACTIVITY IRM LLC (BM) 2008-09-18 WO disclosed
WO-2008112674-A1 COMPOUNDS AND COMPOSITIONS AS INHIBITORS OF CANNABINOID RECEPTOR 1 ACTIVITY IRM LLC (BM) 2008-09-18 WO disclosed