SCHEMBL474386

SCHEMBL474386

COC(=O)c1ccc(-c2ccc(C(C)C(O)(c3ccc(=O)n4ccccc34)C(F)(F)F)cc2)c(Cl)c1F

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDK2 Q15119 1/20 0.36
MAPT P10636 5/20 0.33
MEN1 O00255 4/20 0.33
KMT2A Q03164 4/20 0.33
ALDH1A1 P00352 4/20 0.33
PPARG P37231 2/20 0.33
NCOR2 Q9Y618 2/20 0.33
KDM4E B2RXH2 2/20 0.33
MAPK1 P28482 1/20 0.33
L3MBTL1 Q9Y468 1/20 0.33
NR2E3 Q9Y5X4 1/20 0.33
IDO1 P14902 1/20 0.32
SLC6A4 P31645 2/20 0.32
SLC6A3 Q01959 2/20 0.32
USP2 O75604 1/20 0.31
TDP1 Q9NUW8 2/20 0.31
LMNA P02545 1/20 0.31
NPSR1 Q6W5P4 1/20 0.31
GPR55 Q9Y2T6 1/20 0.31
RECQL P46063 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12163881 0.81 PDK2 (0.36) PDK2MAPTMEN1KMT2AALDH1A1
SCHEMBL474577 0.81 PDK2 (0.36) PDK2MAPTMEN1KMT2AALDH1A1
SCHEMBL474382 0.76 BDKRB1 (0.41)
SCHEMBL474413 0.73 RORC (0.42) PDK2PPARGRORC
SCHEMBL15520363 0.73 NR3C2 (0.33) L3MBTL1RORC
SCHEMBL15520819 0.70 RORC (0.32) PPARGRORC
SCHEMBL473838 0.67 OPRM1 (0.32)
SCHEMBL474580 0.61 AKR1C3 (0.38)
SCHEMBL9338362 0.59 SLC6A4 (0.56) MAPTMEN1KMT2AALDH1A1PPARG
SCHEMBL9335009 0.59 SLC6A4 (0.56) MAPTMEN1KMT2AALDH1A1PPARG

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2411365-A1 2,3-DIARYL- OR HETEROARYL-SUBSTITUTED 1,1,1-TRIFLUORO-2-HYDROXYPROPYL COMPOUNDS F. Hoffmann-La Roche AG (CH) 2012-02-01 EP disclosed
WO-2010108903-A1 2,3-DIARYL- OR HETEROARYL-SUBSTITUTED 1,1,1-TRIFLUORO-2-HYDROXYPROPYL COMPOUNDS F. HOFFMANN-LA ROCHE AG (CH) 2010-09-30 WO disclosed