SCHEMBL9338362

SCHEMBL9338362

COC(=O)c1cc(-c2ccc(Cl)cc2)c(=O)n2ccccc12

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SLC6A4 P31645 1/20 0.56
SLC6A3 Q01959 1/20 0.56
ALDH1A1 P00352 7/20 0.49
KDM4E B2RXH2 6/20 0.49
GAA P10253 2/20 0.49
HPGD P15428 2/20 0.49
GLA P06280 1/20 0.49
KMT2A Q03164 6/20 0.48
MAPT P10636 6/20 0.48
MEN1 O00255 5/20 0.48
USP2 O75604 1/20 0.48
TDP1 Q9NUW8 2/20 0.47
NPSR1 Q6W5P4 2/20 0.47
PPARG P37231 2/20 0.47
NCOR2 Q9Y618 2/20 0.47
LMNA P02545 1/20 0.47
GPR55 Q9Y2T6 1/20 0.47
RECQL P46063 1/20 0.46
RXFP1 Q9HBX9 1/20 0.46
GABRA1 P14867 3/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8173738 0.90 GABRA1 (0.56) ALDH1A1KDM4EGAAHPGDGLA
SCHEMBL9335009 0.88 SLC6A4 (0.56) SLC6A4SLC6A3ALDH1A1KDM4EGAA
SCHEMBL9337598 0.81 MAPT (0.47) SLC6A4SLC6A3ALDH1A1KDM4EGAA
SCHEMBL27273711 0.79 ALDH1A1 (0.50) SLC6A4SLC6A3ALDH1A1KDM4EGAA
SCHEMBL10361534 0.79 KDM4E (0.70) ALDH1A1KDM4EGAAHPGDGLA
SCHEMBL8179828 0.78 MAPT (0.47) ALDH1A1KDM4EGAAHPGDGLA
SCHEMBL10362797 0.78 FNTA (0.53) ALDH1A1KDM4EGAAHPGDGLA
SCHEMBL16467778 0.74 MAPT (0.48) SLC6A4SLC6A3ALDH1A1KDM4EGAA
SCHEMBL8167032 0.73 GABRA1 (0.46) SLC6A4SLC6A3ALDH1A1KDM4EGAA
SCHEMBL24304134 0.71 TP53 (0.63) ALDH1A1KDM4EGAAHPGDGLA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5321021-A Tricyclic pyridine derivatives HOFFMANN-LA ROCHE INC. (US) 1994-06-14 US disclosed
US-5036066-A Muscle relaxants, anxiolytic agents, anticonvulsants HOFFMANN-LA ROCHE INC. (US) 1991-07-30 US disclosed
US-4889848-A 4-OXO-4H-BENZO(A)QUINOLIZINES; MUSCLE RELAXANTS; SEDATIVES; ANTICONVULSANTS; ANXIOLYTIC AGENTS HOFFMANN-LA ROCHE INC. (US) 1989-12-26 US disclosed
US-4735940-A Tricyclic pyridine derivatives and pharmaceutical compositions HOFFMANN-LA ROCHE INC. (US) 1988-04-05 US disclosed