SCHEMBL474431

SCHEMBL474431

COC(=O)c1ccc(-c2ccccc2)c(C(C)C(O)(c2ccc3c(c2)NC(=O)CO3)C(F)(F)F)c1

nearest known ligand 0.48

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
TRPV1 Q8NER1 3/20 0.41
GAA P10253 1/20 0.40
ALDH1A1 P00352 5/20 0.40
MAPK1 P28482 1/20 0.40
NR3C2 P08235 5/20 0.39
NR3C1 P04150 2/20 0.39
LMNA P02545 1/20 0.39
MAPT P10636 3/20 0.39
POLB P06746 1/20 0.39
KDM4E B2RXH2 1/20 0.38
HPGD P15428 1/20 0.38
KMT2A Q03164 1/20 0.38
CASP3 P42574 1/20 0.38
SENP7 Q9BQF6 1/20 0.38
PKM P14618 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL473988 0.92 GAA (0.45) TRPV1GAAALDH1A1MAPK1NR3C2
SCHEMBL474394 0.84 POLB (0.36) ALDH1A1POLBCASP3
SCHEMBL474476 0.76 MAPK14 (0.35) TRPV1POLB
SCHEMBL12163960 0.76 F7 (0.39) TRPV1NR3C2NR3C1CASP3SENP7
SCHEMBL474611 0.76 SMN1; SMN2 (0.35) ALDH1A1POLBKDM4EKMT2ACASP3
SCHEMBL474251 0.76 F7 (0.39) TRPV1NR3C2NR3C1CASP3SENP7
SCHEMBL474504 0.76 NR3C2 (0.40) NR3C2NR3C1
SCHEMBL473917 0.75 ALDH1A1 (0.36) ALDH1A1POLBHPGDKMT2A
SCHEMBL474658 0.74 SMN1; SMN2 (0.36) ALDH1A1POLBKMT2ACASP3
SCHEMBL15520270 0.73 NR3C2 (0.38) TRPV1ALDH1A1NR3C2NR3C1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2411365-A1 2,3-DIARYL- OR HETEROARYL-SUBSTITUTED 1,1,1-TRIFLUORO-2-HYDROXYPROPYL COMPOUNDS F. Hoffmann-La Roche AG (CH) 2012-02-01 EP disclosed