SCHEMBL474476

SCHEMBL474476

COC(=O)c1ccc(-c2ccccc2)c(C(C)C(O)(c2cc3c(cc2F)OCC(=O)N3C)C(F)(F)F)c1

nearest known ligand 0.35

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
MAPK14 Q16539 3/20 0.35
MAP3K5 Q99683 1/20 0.35
POLB P06746 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
USP30 Q70CQ3 1/20 0.34
EGFR P00533 1/20 0.33
PTGER3 P43115 1/20 0.33
PTGS2 P35354 1/20 0.33
TRPV1 Q8NER1 4/20 0.32
CYP11B1 P15538 1/20 0.32
CYP11B2 P19099 1/20 0.32
GPR55 Q9Y2T6 1/20 0.32
CHRM2 P08172 1/20 0.31
CHRM4 P08173 1/20 0.31
CHRM5 P08912 1/20 0.31
CHRM1 P11229 1/20 0.31
CHRM3 P20309 1/20 0.31
WDR5 P61964 1/20 0.31
PDK2 Q15119 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL474394 0.88 POLB (0.36) MAPK14POLBSMN1; SMN2USP30EGFR
SCHEMBL474658 0.86 SMN1; SMN2 (0.36) MAPK14POLBSMN1; SMN2EGFRPTGS2
SCHEMBL474611 0.85 SMN1; SMN2 (0.35) MAPK14POLBSMN1; SMN2EGFRPTGS2
SCHEMBL473908 0.80 BDKRB1 (0.41)
SCHEMBL473958 0.80 ALDH1A1 (0.37) POLBUSP30PTGER3CYP11B1CYP11B2
SCHEMBL474379 0.78 MAP3K5 (0.36) MAP3K5USP30CYP11B1CYP11B2GPR55
SCHEMBL12164119 0.78 MAP3K5 (0.36) MAP3K5USP30CYP11B1CYP11B2GPR55
SCHEMBL474375 0.78 ALDH1A1 (0.37)
SCHEMBL474455 0.76 ALDH1A1 (0.34)
SCHEMBL474073 0.76 MAP3K5 (0.34) MAP3K5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2411365-A1 2,3-DIARYL- OR HETEROARYL-SUBSTITUTED 1,1,1-TRIFLUORO-2-HYDROXYPROPYL COMPOUNDS F. Hoffmann-La Roche AG (CH) 2012-02-01 EP disclosed