SCHEMBL4744476

SCHEMBL4744476

Cc1oc(-c2ccc(C(F)(F)F)cc2)nc1COc1cccc(CN2CCCCC2C(=O)O)c1

nearest known ligand 0.55

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
PPARG P37231 9/20 0.55
PPARA Q07869 9/20 0.55
CYP2C9 P11712 1/20 0.55
KCNH2 Q12809 1/20 0.55
CD274 Q9NZQ7 3/20 0.55
KDR P35968 1/20 0.50
POLB P06746 1/20 0.50
ALDH1A1 P00352 1/20 0.49
SMN1; SMN2 Q16637 1/20 0.49
PTPN1 P18031 1/20 0.48
PDCD1 Q15116 2/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4744118 1.00 PPARG (0.55) PPARGPPARACYP2C9KCNH2CD274
SCHEMBL4748381 0.98 PPARG (0.56) PPARGPPARACYP2C9KCNH2CD274
SCHEMBL4746251 0.98 PPARG (0.56) PPARGPPARACYP2C9KCNH2CD274
SCHEMBL4744641 0.98 PPARG (0.56) PPARGPPARACYP2C9KCNH2CD274
SCHEMBL4744720 0.93 PPARG (0.52) PPARGPPARACYP2C9KCNH2CD274
SCHEMBL4744723 0.93 PPARG (0.52) PPARGPPARACYP2C9KCNH2CD274
SCHEMBL4744590 0.92 ALDH1A1 (0.61) PPARGPPARACYP2C9KCNH2CD274
SCHEMBL4747847 0.91 CD274 (0.63) PPARGPPARACD274KDRPOLB
SCHEMBL4743927 0.91 CD274 (0.65) PPARGPPARACD274KDRPOLB
SCHEMBL4744001 0.91 CD274 (0.65) PPARGPPARACD274KDRPOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008117982-A1 HETEROCYCLIC CARBOXYLIC ACID DERIVATIVES AND PHARMACEUTICAL COMPOSITION FOR INHIBITING LIPID ACCUMULATION CONTAINING SAME CRYSTAL GENOMICS, INC. (KR) 2008-10-02 WO claimed
WO-2008117982-A1 HETEROCYCLIC CARBOXYLIC ACID DERIVATIVES AND PHARMACEUTICAL COMPOSITION FOR INHIBITING LIPID ACCUMULATION CONTAINING SAME CRYSTAL GENOMICS, INC. (KR) 2008-10-02 WO disclosed