SCHEMBL4744592

SCHEMBL4744592

Cc1oc(-c2ccc(C(F)(F)F)cc2)nc1CCOc1ccc(CN2CCCC[C@@H]2C(=O)O)cc1

nearest known ligand 0.55

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
PPARG P37231 16/20 0.55
PPARA Q07869 12/20 0.55
KDM4E B2RXH2 1/20 0.51
ALDH1A1 P00352 1/20 0.51
CYP2C9 P11712 3/20 0.48
CYP2C19 P33261 1/20 0.48
CYP3A4 P08684 1/20 0.48
KCNH2 Q12809 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4744029 1.00 PPARG (0.55) PPARGPPARAKDM4EALDH1A1CYP2C9
SCHEMBL4744028 0.98 PPARG (0.56) PPARGPPARACYP2C9CYP2C19CYP3A4
SCHEMBL4748056 0.98 PPARG (0.56) PPARGPPARACYP2C9CYP2C19CYP3A4
SCHEMBL4744011 0.94 PPARG (0.57) PPARGPPARACYP2C9CYP2C19CYP3A4
SCHEMBL4747359 0.94 PPARG (0.57) PPARGPPARACYP2C9CYP2C19CYP3A4
SCHEMBL4744563 0.93 KDM4E (0.52) PPARGPPARAKDM4EALDH1A1CYP2C9
SCHEMBL4744570 0.93 KDM4E (0.52) PPARGPPARAKDM4EALDH1A1CYP2C9
SCHEMBL4748206 0.92 KDM4E (0.54) PPARGPPARAKDM4EALDH1A1
SCHEMBL4748204 0.92 KDM4E (0.54) PPARGPPARAKDM4EALDH1A1
SCHEMBL4746231 0.92 ALDH1A1 (0.65) PPARGPPARAKDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008117982-A1 HETEROCYCLIC CARBOXYLIC ACID DERIVATIVES AND PHARMACEUTICAL COMPOSITION FOR INHIBITING LIPID ACCUMULATION CONTAINING SAME CRYSTAL GENOMICS, INC. (KR) 2008-10-02 WO claimed
WO-2008117982-A1 HETEROCYCLIC CARBOXYLIC ACID DERIVATIVES AND PHARMACEUTICAL COMPOSITION FOR INHIBITING LIPID ACCUMULATION CONTAINING SAME CRYSTAL GENOMICS, INC. (KR) 2008-10-02 WO disclosed