SCHEMBL4745366

SCHEMBL4745366

CC(C)NC(=O)CN1CCN(CCCCCOc2ccc(C(=O)c3ccc(Cl)c(Cl)c3)cc2)CC1

nearest known ligand 0.53

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
HRH4 Q9H3N8 1/20 0.53
HRH3 Q9Y5N1 7/20 0.49
KDM4E B2RXH2 4/20 0.48
ALDH1A1 P00352 3/20 0.48
SMN1; SMN2 Q16637 2/20 0.48
POLB P06746 1/20 0.48
HTR1A P08908 1/20 0.47
DRD2 P14416 1/20 0.47
HTR2A P28223 1/20 0.47
BCHE P06276 3/20 0.46
ACHE P22303 3/20 0.46
HRH2 P25021 2/20 0.46
HRH1 P35367 2/20 0.46
AVPR1B P47901 1/20 0.46
MEN1 O00255 1/20 0.46
KMT2A Q03164 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4743111 0.90 HRH3 (0.56) HRH4HRH3HRH1MEN1KMT2A
SCHEMBL4743288 0.90 HRH3 (0.56) HRH4HRH3HRH1MEN1KMT2A
SCHEMBL4743293 0.89 MEN1 (0.56) HRH4HRH3KDM4EALDH1A1DRD2
SCHEMBL4743291 0.86 HRH3 (0.48) HRH4HRH3HTR1ADRD2HTR2A
SCHEMBL4745334 0.85 HRH3 (0.47) HRH4HRH3AVPR1BMEN1KMT2A
SCHEMBL21026135 0.83 HRH3 (0.55) HRH3KDM4EALDH1A1HRH2HRH1
SCHEMBL4744692 0.83 KDM4E (0.51) HRH4HRH3KDM4ESMN1; SMN2POLB
SCHEMBL4746716 0.82 HRH3 (0.58) HRH3MEN1KMT2A
SCHEMBL4745400 0.81 HTR1A (0.50) HRH3HTR1ADRD2HTR2AAVPR1B
SCHEMBL4744719 0.81 HRH3 (0.53) HRH3DRD2MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008107320-A1 PIPERIDINE AND PIPERAZINE DERIVATIVES USED AS ANTI-NEOPLASIC AGENTS OR CELL PROLIFERATION INHIBITORS CEREP (FR) 2008-09-12 WO claimed
WO-2008107320-A1 PIPERIDINE AND PIPERAZINE DERIVATIVES USED AS ANTI-NEOPLASIC AGENTS OR CELL PROLIFERATION INHIBITORS CEREP (FR) 2008-09-12 WO disclosed