SCHEMBL4745543

SCHEMBL4745543

O=C(O)c1ccc(CNCc2ccccc2)cc1

nearest known ligand 0.72

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.72
HDAC8 Q9BY41 2/20 0.70
HDAC6 Q9UBN7 1/20 0.70
SMN1; SMN2 Q16637 3/20 0.62
NPSR1 Q6W5P4 1/20 0.59
KDM4E B2RXH2 1/20 0.59
NR1H4 Q96RI1 3/20 0.59
EPHX2 P34913 2/20 0.59
POLB P06746 1/20 0.59
HPGD P15428 1/20 0.59
HSD17B10 Q99714 1/20 0.59
CTDSP1 Q9GZU7 1/20 0.59
L3MBTL1 Q9Y468 1/20 0.59
KMT2A Q03164 3/20 0.58
HDAC3 O15379 1/20 0.53
HDAC1 Q13547 1/20 0.53
HDAC2 Q92769 1/20 0.53
DAO P14920 1/20 0.52
TSHR P16473 1/20 0.52
NAPRT Q6XQN6 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL28066263 0.98 ALDH1A1 (0.70) ALDH1A1HDAC8HDAC6SMN1; SMN2NPSR1
Benzoic Acid SCHEMBL10942201 0.94 ALDH1A1 (0.63) ALDH1A1HDAC8HDAC6SMN1; SMN2NPSR1
SCHEMBL3503996 0.94 ALDH1A1 (0.81) ALDH1A1HDAC8HDAC6SMN1; SMN2NPSR1
Hydrochloric Acid SCHEMBL15392980 0.91 ALDH1A1 (0.78) ALDH1A1HDAC8HDAC6SMN1; SMN2NPSR1
SCHEMBL20846406 0.90 EPHX2 (0.73) ALDH1A1HDAC8HDAC6SMN1; SMN2NPSR1
4-Methylbenzoic Acid SCHEMBL31121234 0.89 SMN1; SMN2 (0.61) ALDH1A1HDAC8HDAC6SMN1; SMN2KDM4E
SCHEMBL9185931 0.87 ALDH1A1 (0.67) ALDH1A1HDAC8HDAC6KDM4EKMT2A
SCHEMBL2938207 0.85 ALDH1A1 (0.69) ALDH1A1HDAC8HDAC6SMN1; SMN2NPSR1
Bicarbonate SCHEMBL23420914 0.84 HDAC8 (0.64) HDAC8HDAC6SMN1; SMN2KMT2AHDAC3
Bicarbonate SCHEMBL11577277 0.84 HDAC8 (0.64) HDAC8HDAC6SMN1; SMN2KMT2AHDAC3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 10 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2861568-B1 TERTIARY AMINES FOR USE IN THE TREATMENT OF CARDIAC DISORDERS UNIV OSLO (NO) 2019-04-17 EP disclosed
EP-3331864-A2 1,3,4-OXADIAZOLE DERIVATIVE COMPOUNDS AS HISTONE DEACETYLASE 6 INHIBITOR, AND THE PHARMACEUTICAL COMPOSITION COMPRISING THE SAME Chong Kun Dang Pharmaceutical Corp. (KR) 2018-06-13 EP disclosed
US-20080293711-A1 Chemokine receptor modulators METASTATIX, INC. 2008-11-27 US disclosed
US-20080293711-A1 Chemokine receptor modulators METASTATIX, INC. 2008-11-27 US disclosed
US-20080293711-A1 Chemokine receptor modulators METASTATIX, INC. 2008-11-27 US disclosed
US-20080261978-A1 treating or preventing HIV infections, and in treating proliferative disorders such as inhibiting the metastasis of various cancers; 1-(4-((pyridin-2-ylmethylamino)methyl)benzyl)-3-phenylurea METASTATIX, INC. 2008-10-23 US disclosed
US-20080261978-A1 treating or preventing HIV infections, and in treating proliferative disorders such as inhibiting the metastasis of various cancers; 1-(4-((pyridin-2-ylmethylamino)methyl)benzyl)-3-phenylurea METASTATIX, INC. 2008-10-23 US disclosed
WO-2008112156-A1 CHEMOKINE RECEPTOR MODULATORS ALTIRIS THERAPEUTICS (US) 2008-09-18 WO disclosed
WO-2008112156-A1 CHEMOKINE RECEPTOR MODULATORS ALTIRIS THERAPEUTICS (US) 2008-09-18 WO disclosed
WO-2008109154-A1 CHEMOKINE RECEPTOR MODULATORS ALTIRIS THERAPEUTICS, INC. (US) 2008-09-12 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20080261978-A1 treating or preventing HIV infections, and in treating proliferative disorders such as inhibiting the metastasis of various cancers; 1-(4-((pyridin-2-ylmethylamino)methyl)benzyl)-3-phenylurea MKI67, CCNI, CDKN1A ALDH1A1 423/4885HDAC8 2488/4885HDAC6 1192/4885
US-20080293711-A1 Chemokine receptor modulators CCR5, CCL2, CXCR4 ALDH1A1 1359/4885HDAC8 2165/4885HDAC6 1039/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.